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Discovery of Highly Potent and Efficient PROTAC Degraders of Androgen Receptor (AR) by Employing Weak Binding Affinity VHL E3 Ligase Ligands. [electronic resource] by
- Han, Xin
- Zhao, Lijie
- Xiang, Weiguo
- Qin, Chong
- Miao, Bukeyan
- Xu, Tianfeng
- Wang, Mi
- Yang, Chao-Yie
- Chinnaswamy, Krishnapriya
- Stuckey, Jeanne
- Wang, Shaomeng
Producer: 20200622
In:
Journal of medicinal chemistry vol. 62
Availability: No items available.
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5.
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Structure-Based Design of γ-Carboline Analogues as Potent and Specific BET Bromodomain Inhibitors. [electronic resource] by
- Ran, Xu
- Zhao, Yujun
- Liu, Liu
- Bai, Longchuan
- Yang, Chao-Yie
- Zhou, Bing
- Meagher, Jennifer L
- Chinnaswamy, Krishnapriya
- Stuckey, Jeanne A
- Wang, Shaomeng
Producer: 20150914
In:
Journal of medicinal chemistry vol. 58
Availability: No items available.
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Discovery of M-808 as a Highly Potent, Covalent, Small-Molecule Inhibitor of the Menin-MLL Interaction with Strong [electronic resource] by
- Xu, Shilin
- Aguilar, Angelo
- Huang, Liyue
- Xu, Tianfeng
- Zheng, Ke
- McEachern, Donna
- Przybranowski, Sally
- Foster, Caroline
- Zawacki, Kaitlin
- Liu, Zhaomin
- Chinnaswamy, Krishnapriya
- Stuckey, Jeanne
- Wang, Shaomeng
Producer: 20201021
In:
Journal of medicinal chemistry vol. 63
Availability: No items available.
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7.
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Discovery of ARD-69 as a Highly Potent Proteolysis Targeting Chimera (PROTAC) Degrader of Androgen Receptor (AR) for the Treatment of Prostate Cancer. [electronic resource] by
- Han, Xin
- Wang, Chao
- Qin, Chong
- Xiang, Weiguo
- Fernandez-Salas, Ester
- Yang, Chao-Yie
- Wang, Mi
- Zhao, Lijie
- Xu, Tianfeng
- Chinnaswamy, Krishnapriya
- Delproposto, James
- Stuckey, Jeanne
- Wang, Shaomeng
Producer: 20191017
In:
Journal of medicinal chemistry vol. 62
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8.
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Discovery of ERD-308 as a Highly Potent Proteolysis Targeting Chimera (PROTAC) Degrader of Estrogen Receptor (ER). [electronic resource] by
- Hu, Jiantao
- Hu, Biao
- Wang, Mingliang
- Xu, Fuming
- Miao, Bukeyan
- Yang, Chao-Yie
- Wang, Mi
- Liu, Zhaomin
- Hayes, Daniel F
- Chinnaswamy, Krishnapriya
- Delproposto, James
- Stuckey, Jeanne
- Wang, Shaomeng
Producer: 20200303
In:
Journal of medicinal chemistry vol. 62
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9.
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A potent small-molecule inhibitor of the DCN1-UBC12 interaction that selectively blocks cullin 3 neddylation. [electronic resource] by
- Zhou, Haibin
- Lu, Jianfeng
- Liu, Liu
- Bernard, Denzil
- Yang, Chao-Yie
- Fernandez-Salas, Ester
- Chinnaswamy, Krishnapriya
- Layton, Stephanie
- Stuckey, Jeanne
- Yu, Qing
- Zhou, Weihua
- Pan, Zhenqiang
- Sun, Yi
- Wang, Shaomeng
Producer: 20181001
In:
Nature communications vol. 8
Availability: No items available.
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10.
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Design of the First-in-Class, Highly Potent Irreversible Inhibitor Targeting the Menin-MLL Protein-Protein Interaction. [electronic resource] by
- Xu, Shilin
- Aguilar, Angelo
- Xu, Tianfeng
- Zheng, Ke
- Huang, Liyue
- Stuckey, Jeanne
- Chinnaswamy, Krishnapriya
- Bernard, Denzil
- Fernández-Salas, Ester
- Liu, Liu
- Wang, Mi
- McEachern, Donna
- Przybranowski, Sally
- Foster, Caroline
- Wang, Shaomeng
Producer: 20190403
In:
Angewandte Chemie (International ed. in English) vol. 57
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11.
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High-Affinity Peptidomimetic Inhibitors of the DCN1-UBC12 Protein-Protein Interaction. [electronic resource] by
- Zhou, Haibin
- Zhou, Weihua
- Zhou, Bing
- Liu, Liu
- Chern, Ting-Rong
- Chinnaswamy, Krishnapriya
- Lu, Jianfeng
- Bernard, Denzil
- Yang, Chao-Yie
- Li, Shasha
- Wang, Mi
- Stuckey, Jeanne
- Sun, Yi
- Wang, Shaomeng
Producer: 20190503
In:
Journal of medicinal chemistry vol. 61
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12.
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From proteomics to discovery of first-in-class ST2 inhibitors active in vivo. [electronic resource] by
- Ramadan, Abdulraouf M
- Daguindau, Etienne
- Rech, Jason C
- Chinnaswamy, Krishnapriya
- Zhang, Jilu
- Hura, Greg L
- Griesenauer, Brad
- Bolten, Zachary
- Robida, Aaron
- Larsen, Martha
- Stuckey, Jeanne A
- Yang, Chao-Yie
- Paczesny, Sophie
Producer: 20191104
In:
JCI insight vol. 3
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Mechanistic evaluation and transcriptional signature of a glutathione S-transferase omega 1 inhibitor. [electronic resource] by
- Ramkumar, Kavya
- Samanta, Soma
- Kyani, Anahita
- Yang, Suhui
- Tamura, Shuzo
- Ziemke, Elizabeth
- Stuckey, Jeanne A
- Li, Si
- Chinnaswamy, Krishnapriya
- Otake, Hiroyuki
- Debnath, Bikash
- Yarovenko, Vladimir
- Sebolt-Leopold, Judith S
- Ljungman, Mats
- Neamati, Nouri
Producer: 20180910
In:
Nature communications vol. 7
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14.
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CSAR data set release 2012: ligands, affinities, complexes, and docking decoys. [electronic resource] by
- Dunbar, James B
- Smith, Richard D
- Damm-Ganamet, Kelly L
- Ahmed, Aqeel
- Esposito, Emilio Xavier
- Delproposto, James
- Chinnaswamy, Krishnapriya
- Kang, You-Na
- Kubish, Ginger
- Gestwicki, Jason E
- Stuckey, Jeanne A
- Carlson, Heather A
Producer: 20140321
In:
Journal of chemical information and modeling vol. 53
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15.
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Structure-Based Discovery of M-89 as a Highly Potent Inhibitor of the Menin-Mixed Lineage Leukemia (Menin-MLL) Protein-Protein Interaction. [electronic resource] by
- Aguilar, Angelo
- Zheng, Ke
- Xu, Tianfeng
- Xu, Shilin
- Huang, Liyue
- Fernandez-Salas, Ester
- Liu, Liu
- Bernard, Denzil
- Harvey, Kaitlin P
- Foster, Caroline
- McEachern, Donna
- Stuckey, Jeanne
- Chinnaswamy, Krishnapriya
- Delproposto, James
- Kampf, Jeff W
- Wang, Shaomeng
Producer: 20200601
In:
Journal of medicinal chemistry vol. 62
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16.
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CSAR Benchmark Exercise 2013: Evaluation of Results from a Combined Computational Protein Design, Docking, and Scoring/Ranking Challenge. [electronic resource] by
- Smith, Richard D
- Damm-Ganamet, Kelly L
- Dunbar, James B
- Ahmed, Aqeel
- Chinnaswamy, Krishnapriya
- Delproposto, James E
- Kubish, Ginger M
- Tinberg, Christine E
- Khare, Sagar D
- Dou, Jiayi
- Doyle, Lindsey
- Stuckey, Jeanne A
- Baker, David
- Carlson, Heather A
Producer: 20170811
In:
Journal of chemical information and modeling vol. 56
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17.
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A Potent and Selective Small-Molecule Degrader of STAT3 Achieves Complete Tumor Regression In Vivo. [electronic resource] by
- Bai, Longchuan
- Zhou, Haibin
- Xu, Renqi
- Zhao, Yujun
- Chinnaswamy, Krishnapriya
- McEachern, Donna
- Chen, Jianyong
- Yang, Chao-Yie
- Liu, Zhaomin
- Wang, Mi
- Liu, Liu
- Jiang, Hui
- Wen, Bo
- Kumar, Praveen
- Meagher, Jennifer L
- Sun, Duxin
- Stuckey, Jeanne A
- Wang, Shaomeng
Producer: 20200527
In:
Cancer cell vol. 36
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18.
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Structure-Based Discovery of SD-36 as a Potent, Selective, and Efficacious PROTAC Degrader of STAT3 Protein. [electronic resource] by
- Zhou, Haibin
- Bai, Longchuan
- Xu, Renqi
- Zhao, Yujun
- Chen, Jianyong
- McEachern, Donna
- Chinnaswamy, Krishnapriya
- Wen, Bo
- Dai, Lipeng
- Kumar, Praveen
- Yang, Chao-Yie
- Liu, Zhaomin
- Wang, Mi
- Liu, Liu
- Meagher, Jennifer L
- Yi, Han
- Sun, Duxin
- Stuckey, Jeanne A
- Wang, Shaomeng
Producer: 20200622
In:
Journal of medicinal chemistry vol. 62
Availability: No items available.
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19.
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Changing the Apoptosis Pathway through Evolutionary Protein Design. [electronic resource] by
- Shultis, David
- Mitra, Pralay
- Huang, Xiaoqiang
- Johnson, Jarrett
- Khattak, Naureen Aslam
- Gray, Felicia
- Piper, Clint
- Czajka, Jeff
- Hansen, Logan
- Wan, Bingbing
- Chinnaswamy, Krishnapriya
- Liu, Liu
- Wang, Mi
- Pan, Jingxi
- Stuckey, Jeanne
- Cierpicki, Tomasz
- Borchers, Christoph H
- Wang, Shaomeng
- Lei, Ming
- Zhang, Yang
Producer: 20200302
In:
Journal of molecular biology vol. 431
Availability: No items available.
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20.
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Discovery and Characterization of 2,5-Substituted Benzoic Acid Dual Inhibitors of the Anti-apoptotic Mcl-1 and Bfl-1 Proteins. [electronic resource] by
- Kump, Karson J
- Miao, Lei
- Mady, Ahmed S A
- Ansari, Nurul H
- Shrestha, Uttar K
- Yang, Yuting
- Pal, Mohan
- Liao, Chenzhong
- Perdih, Andrej
- Abulwerdi, Fardokht A
- Chinnaswamy, Krishnapriya
- Meagher, Jennifer L
- Carlson, Jacob M
- Khanna, May
- Stuckey, Jeanne A
- Nikolovska-Coleska, Zaneta
Producer: 20200831
In:
Journal of medicinal chemistry vol. 63
Availability: No items available.
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