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Macrocyclic ureas as potent and selective Chk1 inhibitors: an improved synthesis, kinome profiling, structure-activity relationships, and preliminary pharmacokinetics. [electronic resource] by
- Tao, Zhi-Fu
- Chen, Zehan
- Bui, Mai-Ha
- Kovar, Peter
- Johnson, Eric
- Bouska, Jennifer
- Zhang, Haiying
- Rosenberg, Saul
- Sowin, Thomas
- Lin, Nan-Horng
Producer: 20080303
In:
Bioorganic & medicinal chemistry letters vol. 17
Availability: No items available.
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9.
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Synthesis and in-vitro biological activity of macrocyclic urea Chk1 inhibitors. [electronic resource] by
- Li, Gaoquan
- Tao, Zhi-Fu
- Tong, Yunsong
- Przytulinska, Magdalena K
- Kovar, Peter
- Merta, Philip
- Chen, Zehan
- Zhang, Haiying
- Sowin, Thomas
- Rosenberg, Saul H
- Lin, Nan-Horng
Producer: 20080303
In:
Bioorganic & medicinal chemistry letters vol. 17
Availability: No items available.
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10.
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Synthesis and biological evaluation of 4'-(6,7-disubstituted-2,4-dihydro-indeno[1,2-c]pyrazol-3-yl)-biphenyl-4-ol as potent Chk1 inhibitors. [electronic resource] by
- Tao, Zhi-Fu
- Li, Gaoquan
- Tong, Yunsong
- Chen, Zehan
- Merta, Philip
- Kovar, Peter
- Zhang, Haiying
- Rosenberg, Saul H
- Sham, Hing L
- Sowin, Thomas J
- Lin, Nan-Horng
Producer: 20071001
In:
Bioorganic & medicinal chemistry letters vol. 17
Availability: No items available.
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11.
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1-(5-Chloro-2-alkoxyphenyl)-3-(5-cyanopyrazin-2-yl)ureas [correction of cyanopyrazi] as potent and selective inhibitors of Chk1 kinase: synthesis, preliminary SAR, and biological activities. [electronic resource] by
- Wang, Gary T
- Li, Gaoquan
- Mantei, Robert A
- Chen, Zehan
- Kovar, Peter
- Gu, Wendy
- Xiao, Zhan
- Zhang, Haiying
- Sham, Hing L
- Sowin, Thomas
- Rosenberg, Saul H
- Lin, Nan-Horng
Producer: 20050603
In:
Journal of medicinal chemistry vol. 48
Availability: No items available.
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12.
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Synthesis of 1H-pyridin-2-one derivatives as potent and selective farnesyltransferase inhibitors. [electronic resource] by
- Wang, Le
- Lin, Nan-Horng
- Li, Qun
- Henry, Rodger F
- Zhang, Haiying
- Cohen, Jerome
- Gu, Wen-Zhen
- Marsh, Kennan C
- Bauch, Joy L
- Rosenberg, Saul H
- Sham, Hing L
Producer: 20050307
In:
Bioorganic & medicinal chemistry letters vol. 14
Availability: No items available.
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13.
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Design, synthesis, and activity of achiral analogs of 2-quinolones and indoles as non-thiol farnesyltransferase inhibitors. [electronic resource] by
- Li, Qun
- Woods, Keith W
- Wang, Weibo
- Lin, Nan-Horng
- Claiborne, Akiyo
- Gu, Wen-zhen
- Cohen, Jerry
- Stoll, Vincent S
- Hutchins, Charles
- Frost, David
- Rosenberg, Saul H
- Sham, Hing L
Producer: 20050818
In:
Bioorganic & medicinal chemistry letters vol. 15
Availability: No items available.
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14.
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Phenyl Glycolipids with Different Glycosyl Groups Exhibit Marked Differences in Murine and Human iNKT Cell Activation. [electronic resource] by
- Wu, Tai-Na
- Lin, Kun-Hsien
- Wu, Ying-Ta
- Huang, Jing-Rong
- Hung, Jung-Tung
- Wu, Jen-Chine
- Chen, Chien-Yu
- Chu, Kuo-Ching
- Lin, Nan-Horng
- Yu, Alice L
- Wong, Chi-Huey
Producer: 20170310
In:
ACS chemical biology vol. 11
Availability: No items available.
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15.
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Structure-based design, synthesis, and biological evaluation of potent and selective macrocyclic checkpoint kinase 1 inhibitors. [electronic resource] by
- Tao, Zhi-Fu
- Wang, Le
- Stewart, Kent D
- Chen, Zehan
- Gu, Wendy
- Bui, Mai-Ha
- Merta, Philip
- Zhang, Haiying
- Kovar, Peter
- Johnson, Eric
- Park, Chang
- Judge, Russell
- Rosenberg, Saul
- Sowin, Thomas
- Lin, Nan-Horng
Producer: 20070514
In:
Journal of medicinal chemistry vol. 50
Availability: No items available.
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16.
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Investigation of novel 7,8-disubstituted-5,10-dihydro-dibenzo[b,e][1,4]diazepin-11-ones as potent Chk1 inhibitors. [electronic resource] by
- Hasvold, Lisa A
- Wang, Le
- Przytulinska, Magdalena
- Xiao, Zhan
- Chen, Zehan
- Gu, Wen-Zhen
- Merta, Philip J
- Xue, John
- Kovar, Peter
- Zhang, Haiying
- Park, Chang
- Sowin, Thomas J
- Rosenberg, Saul H
- Lin, Nan-Horng
Producer: 20080708
In:
Bioorganic & medicinal chemistry letters vol. 18
Availability: No items available.
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17.
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Isoxazolo[3,4-b]quinoline-3,4(1H,9H)-diones as unique, potent and selective inhibitors for Pim-1 and Pim-2 kinases: chemistry, biological activities, and molecular modeling. [electronic resource] by
- Tong, Yunsong
- Stewart, Kent D
- Thomas, Sheela
- Przytulinska, Magdalena
- Johnson, Eric F
- Klinghofer, Vered
- Leverson, Joel
- McCall, Owen
- Soni, Niru B
- Luo, Yan
- Lin, Nan-horng
- Sowin, Thomas J
- Giranda, Vincent L
- Penning, Thomas D
Producer: 20081030
In:
Bioorganic & medicinal chemistry letters vol. 18
Availability: No items available.
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18.
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Discovery of 4'-(1,4-dihydro-indeno[1,2-c]pyrazol-3-yl)-benzonitriles and 4'-(1,4-dihydro-indeno[1,2-c]pyrazol-3-yl)-pyridine-2'-carbonitriles as potent checkpoint kinase 1 (Chk1) inhibitors. [electronic resource] by
- Tao, Zhi-Fu
- Li, Gaoquan
- Tong, Yunsong
- Stewart, Kent D
- Chen, Zehan
- Bui, Mai-Ha
- Merta, Philip
- Park, Chang
- Kovar, Peter
- Zhang, Haiying
- Sham, Hing L
- Rosenberg, Saul H
- Sowin, Thomas J
- Lin, Nan-Horng
Producer: 20080205
In:
Bioorganic & medicinal chemistry letters vol. 17
Availability: No items available.
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19.
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Discovery of potent imidazole and cyanophenyl containing farnesyltransferase inhibitors with improved oral bioavailability. [electronic resource] by
- Tong, Yunsong
- Lin, Nan-Horng
- Wang, Le
- Hasvold, Lisa
- Wang, Weibo
- Leonard, Nicholas
- Li, Tongmei
- Li, Qun
- Cohen, Jerry
- Gu, Wen-Zhen
- Zhang, Haiying
- Stoll, Vincent
- Bauch, Joy
- Marsh, Kennan
- Rosenberg, Saul H
- Sham, Hing L
Producer: 20040106
In:
Bioorganic & medicinal chemistry letters vol. 13
Availability: No items available.
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20.
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Unprecedented Role of Hybrid N-Glycans as Ligands for HIV-1 Broadly Neutralizing Antibodies. [electronic resource] by
- Shivatare, Vidya S
- Shivatare, Sachin S
- Lee, Chang-Chun David
- Liang, Chi-Hui
- Liao, Kuo-Shiang
- Cheng, Yang-Yu
- Saidachary, Gannerla
- Wu, Chung-Yi
- Lin, Nan-Horng
- Kwong, Peter D
- Burton, Dennis R
- Wu, Chung-Yi
- Wong, Chi-Huey
Producer: 20180709
In:
Journal of the American Chemical Society vol. 140
Availability: No items available.
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