Isoxazolo[3,4-b]quinoline-3,4(1H,9H)-diones as unique, potent and selective inhibitors for Pim-1 and Pim-2 kinases: chemistry, biological activities, and molecular modeling. [electronic resource]
Producer: 20081030Description: 5206-8 p. digitalISSN:- 1464-3405
- Combinatorial Chemistry Techniques
- Crystallography, X-Ray
- Humans
- Isoxazoles -- chemical synthesis
- Models, Molecular
- Molecular Conformation
- Molecular Structure
- Protein Serine-Threonine Kinases -- antagonists & inhibitors
- Proto-Oncogene Proteins -- antagonists & inhibitors
- Proto-Oncogene Proteins c-pim-1 -- antagonists & inhibitors
- Quinolines -- chemical synthesis
- Structure-Activity Relationship
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Publication Type: Journal Article
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