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	1.	A new class of selective, non-basic 5-HT2A receptor antagonists. [electronic resource] by Ladduwahetty, Tammy Boase, Amanda L Mitchinson, Andrew Quin, Caroline Patel, Smita Chapman, Kerry MacLeod, Angus M Producer: 20060816 In: Bioorganic & medicinal chemistry letters vol. 16 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	2.	2,5-Disubstituted pyridines: the discovery of a novel series of 5-HT2A ligands. [electronic resource] by Wilson, Kevin J van Niel, Monique B Cooper, Laura Bloomfield, Dawn O'Connor, Desmond Fish, L Rebecca MacLeod, Angus M Producer: 20070724 In: Bioorganic & medicinal chemistry letters vol. 17 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	3.	3,4-Dihydronaphthalen-1(2H)-ones: novel ligands for the benzodiazepine site of alpha5-containing GABAA receptors. [electronic resource] by Szekeres, Helen J Atack, John R Chambers, Mark S Cook, Susan M Macaulay, Alison J Pillai, Gopalan V MacLeod, Angus M Producer: 20050104 In: Bioorganic & medicinal chemistry letters vol. 14 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	4.	Identification of a series of compounds with potent antiviral activity for the treatment of enterovirus infections. [electronic resource] by MacLeod, Angus M Mitchell, Dale R Palmer, Nicholas J Van de Poël, Hervé Conrath, Katja Andrews, Martin Leyssen, Pieter Neyts, Johan Producer: 20140605 In: ACS medicinal chemistry letters vol. 4 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	5.	Non-basic ligands for aminergic GPCRs: the discovery and development diaryl sulfones as selective, orally bioavailable 5-HT2A receptor antagonists for the treatment of sleep disorders. [electronic resource] by Ladduwahetty, Tammy Gilligan, Myra Humphries, Alexander Merchant, Kevin J Fish, Rebecca McAlister, George Ivarsson, Magnus Dominguez, Maria O'Connor, Desmond MacLeod, Angus M Producer: 20100913 In: Bioorganic & medicinal chemistry letters vol. 20 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	6.	An orally bioavailable, functionally selective inverse agonist at the benzodiazepine site of GABAA alpha5 receptors with cognition enhancing properties. [electronic resource] by Chambers, Mark S Atack, John R Carling, Robert W Collinson, Neil Cook, Susan M Dawson, Gerard R Ferris, Pushpindar Hobbs, Sarah C O'connor, Desmond Marshall, George Rycroft, W Macleod, Angus M Producer: 20050103 In: Journal of medicinal chemistry vol. 47 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	7.	4-Fluorosulfonylpiperidines: selective 5-HT2A ligands for the treatment of insomnia. [electronic resource] by Fish, L Rebecca Gilligan, Myra T Humphries, Alexander C Ivarsson, Magnus Ladduwahetty, Tammy Merchant, Kevin J O'Connor, Desmond Patel, Smita Philipps, Elisabeth Vargas, Hugo M Hutson, Peter H MacLeod, Angus M Producer: 20051205 In: Bioorganic & medicinal chemistry letters vol. 15 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	8.	Identification of a novel, selective GABA(A) alpha5 receptor inverse agonist which enhances cognition. [electronic resource] by Chambers, Mark S Atack, John R Broughton, Howard B Collinson, Neil Cook, Susan Dawson, Gerard R Hobbs, Sarah C Marshall, George Maubach, Karen A Pillai, Goplan V Reeve, Austin J MacLeod, Angus M Producer: 20030623 In: Journal of medicinal chemistry vol. 46 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	9.	6,7-Dihydro-2-benzothiophen-4(5H)-ones: a novel class of GABA-A alpha5 receptor inverse agonists. [electronic resource] by Chambers, Mark S Atack, John R Bromidge, Frances A Broughton, Howard B Cook, Susan Dawson, Gerard R Hobbs, Sarah C Maubach, Karen A Reeve, Austin J Seabrook, Guy R Wafford, Keith MacLeod, Angus M Producer: 20020426 In: Journal of medicinal chemistry vol. 45 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	10.	Pharmacokinetics and metabolism studies on (3-tert-butyl-7-(5-methylisoxazol-3-yl)-2-(1-methyl-1H-1,2,4-triazol-5-ylmethoxy) pyrazolo[1,5-d][1,2,4]triazine, a functionally selective GABA(A) alpha5 inverse agonist for cognitive dysfunction. [electronic resource] by Jones, Philip Atack, John R Braun, Matthew P Cato, Brian P Chambers, Mark S O'Connor, Desmond Cook, Susan M Hobbs, Sarah C Maxey, Robert Szekeres, Helen J Szeto, Nicola Wafford, Keith A MacLeod, Angus M Producer: 20060427 In: Bioorganic & medicinal chemistry letters vol. 16 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	11.	A new pyridazine series of GABAA alpha5 ligands. [electronic resource] by van Niel, Monique B Wilson, Kevin Adkins, Charles H Atack, John R Castro, José L Clarke, Dawn E Fletcher, Stephen Gerhard, Ute Mackey, Mark M Malpas, Sallie Maubach, Karen Newman, Robert O'Connor, Desmond Pillai, Gopalan V Simpson, Peter B Thomas, Steven R MacLeod, Angus M Producer: 20051108 In: Journal of medicinal chemistry vol. 48 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	12.	Selective, orally active gamma-aminobutyric acidA alpha5 receptor inverse agonists as cognition enhancers. [electronic resource] by Sternfeld, Francine Carling, Robert W Jelley, Richard A Ladduwahetty, Tamara Merchant, Kevin J Moore, Kevin W Reeve, Austin J Street, Leslie J O'Connor, Desmond Sohal, Bindi Atack, John R Cook, Susan Seabrook, Guy Wafford, Keith Tattersall, F David Collinson, Neil Dawson, Gerard R Castro, José L MacLeod, Angus M Producer: 20040520 In: Journal of medicinal chemistry vol. 47 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	13.	4-(Phenylsulfonyl)piperidines: novel, selective, and bioavailable 5-HT(2A) receptor antagonists. [electronic resource] by Fletcher, Stephen R Burkamp, Frank Blurton, Peter Cheng, Susan K F Clarkson, Robert O'Connor, Desmond Spinks, Daniel Tudge, Matthew van Niel, Monique B Patel, Smita Chapman, Kerry Marwood, Rose Shepheard, Sara Bentley, Graham Cook, Gina P Bristow, Linda J Castro, Jose L Hutson, Peter H MacLeod, Angus M Producer: 20020207 In: Journal of medicinal chemistry vol. 45 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	14.	A novel, broad-spectrum inhibitor of enterovirus replication that targets host cell factor phosphatidylinositol 4-kinase IIIβ. [electronic resource] by van der Schaar, Hilde M Leyssen, Pieter Thibaut, Hendrik J de Palma, Armando van der Linden, Lonneke Lanke, Kjerstin H W Lacroix, Céline Verbeken, Erik Conrath, Katja Macleod, Angus M Mitchell, Dale R Palmer, Nicholas J van de Poël, Hervé Andrews, Martin Neyts, Johan van Kuppeveld, Frank J M Producer: 20140409 In: Antimicrobial agents and chemotherapy vol. 57 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	15.	Identification of an Orally Bioavailable, Potent, and Selective Inhibitor of GlyT1. [electronic resource] by Blackaby, Wesley P Lewis, Richard T Thomson, Joanne L Jennings, Andrew S R Goodacre, Simon C Street, Leslie J MacLeod, Angus M Pike, Andrew Wood, Suzanne Thomas, Steve Brown, Terry A Smith, Alison Pillai, Gopalan Almond, Sarah Guscott, Martin R Burns, H Donald Eng, Waisi Ryan, Christine Cook, Jacquelynn Hamill, Terence G Producer: 20140605 In: ACS medicinal chemistry letters vol. 1 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	16.	Synthesis and biological evaluation of 3-heterocyclyl-7,8,9,10-tetrahydro-(7,10-ethano)-1,2,4-triazolo[3,4-a]phthalazines and analogues as subtype-selective inverse agonists for the GABA(A)alpha5 benzodiazepine binding site. [electronic resource] by Street, Leslie J Sternfeld, Francine Jelley, Richard A Reeve, Austin J Carling, Robert W Moore, Kevin W McKernan, Ruth M Sohal, Bindi Cook, Susan Pike, Andrew Dawson, Gerard R Bromidge, Frances A Wafford, Keith A Seabrook, Guy R Thompson, Sally A Marshall, George Pillai, Goplan V Castro, José L Atack, John R MacLeod, Angus M Producer: 20040802 In: Journal of medicinal chemistry vol. 47 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	17.	A small molecule mitigates hearing loss in a mouse model of Usher syndrome III. [electronic resource] by Alagramam, Kumar N Gopal, Suhasini R Geng, Ruishuang Chen, Daniel H-C Nemet, Ina Lee, Richard Tian, Guilian Miyagi, Masaru Malagu, Karine F Lock, Christopher J Esmieu, William R K Owens, Andrew P Lindsay, Nicola A Ouwehand, Krista Albertus, Faywell Fischer, David F Bürli, Roland W MacLeod, Angus M Harte, William E Palczewski, Krzysztof Imanishi, Yoshikazu Producer: 20170502 In: Nature chemical biology vol. 12 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	18.	In vitro and in vivo properties of 3-tert-butyl-7-(5-methylisoxazol-3-yl)-2-(1-methyl-1H-1,2,4-triazol-5-ylmethoxy)-pyrazolo[1,5-d]-[1,2,4]triazine (MRK-016), a GABAA receptor alpha5 subtype-selective inverse agonist. [electronic resource] by Atack, John R Maubach, Karen A Wafford, Keith A O'Connor, Desmond Rodrigues, A David Evans, David C Tattersall, F David Chambers, Mark S MacLeod, Angus M Eng, Wai-Si Ryan, Christine Hostetler, Eric Sanabria, Sandra M Gibson, Raymond E Krause, Stephen Burns, H Donald Hargreaves, Richard J Agrawal, Nancy G B McKernan, Ruth M Murphy, M Gail Gingrich, Kevin Dawson, Gerard R Musson, Donald G Petty, Kevin J Producer: 20091130 In: The Journal of pharmacology and experimental therapeutics vol. 331 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)