An orally bioavailable, functionally selective inverse agonist at the benzodiazepine site of GABAA alpha5 receptors with cognition enhancing properties. [electronic resource]
Producer: 20050103Description: 5829-32 p. digitalISSN:- 0022-2623
- Administration, Oral
- Animals
- Binding Sites
- Biological Availability
- Cognition -- drug effects
- Dogs
- GABA-A Receptor Agonists
- Isoxazoles -- adverse effects
- Maze Learning -- drug effects
- Mice
- Nootropic Agents -- adverse effects
- Patch-Clamp Techniques
- Protein Subunits
- Radioligand Assay
- Rats
- Receptors, GABA-A -- metabolism
- Triazines -- adverse effects
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Publication Type: Journal Article
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