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N-substituted azaindoles as potent inhibitors of Cdc7 kinase. [electronic resource] by
- Bryan, Marian C
- Falsey, James R
- Frohn, Mike
- Reichelt, Andreas
- Yao, Guomin
- Bartberger, Michael D
- Bailis, Julie M
- Zalameda, Leeanne
- Miguel, Tisha San
- Doherty, Elizabeth M
- Allen, John G
Producer: 20130930
In:
Bioorganic & medicinal chemistry letters vol. 23
Availability: No items available.
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8.
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Design and synthesis of peripherally restricted transient receptor potential vanilloid 1 (TRPV1) antagonists. [electronic resource] by
- Tamayo, Nuria
- Liao, Hongyu
- Stec, Markian M
- Wang, Xianghong
- Chakrabarti, Partha
- Retz, Dan
- Doherty, Elizabeth M
- Surapaneni, Sekhar
- Tamir, Rami
- Bannon, Anthony W
- Gavva, Narender R
- Norman, Mark H
Producer: 20080709
In:
Journal of medicinal chemistry vol. 51
Availability: No items available.
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9.
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Structure-guided Discovery of Dual-recognition Chemibodies. [electronic resource] by
- Cheng, Alan C
- Doherty, Elizabeth M
- Johnstone, Sheree
- DiMauro, Erin F
- Dao, Jennifer
- Luthra, Abhinav
- Ye, Jay
- Tang, Jie
- Nixey, Thomas
- Min, Xiaoshan
- Tagari, Philip
- Miranda, Les P
- Wang, Zhulun
Producer: 20191015
In:
Scientific reports vol. 8
Availability: No items available.
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10.
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Synthesis and evaluation of thiazole carboxamides as vanilloid receptor 1 (TRPV1) antagonists. [electronic resource] by
- Xi, Ning
- Bo, Yunxin
- Doherty, Elizabeth M
- Fotsch, Christopher
- Gavva, Narender R
- Han, Nianhe
- Hungate, Randall W
- Klionsky, Lana
- Liu, Qingyian
- Tamir, Rami
- Xu, Shimin
- Treanor, James J S
- Norman, Mark H
Producer: 20060123
In:
Bioorganic & medicinal chemistry letters vol. 15
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11.
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Design of a new peptidomimetic agonist for the melanocortin receptors based on the solution structure of the peptide ligand, Ac-Nle-cyclo[Asp-Pro-DPhe-Arg-Trp-Lys]-NH(2). [electronic resource] by
- Fotsch, Christopher
- Smith, Duncan M
- Adams, Jeffrey A
- Cheetham, Janet
- Croghan, Michael
- Doherty, Elizabeth M
- Hale, Clarence
- Jarosinski, Mark A
- Kelly, Michael G
- Norman, Mark H
- Tamayo, Nuria A
- Xi, Ning
- Baumgartner, James W
Producer: 20040227
In:
Bioorganic & medicinal chemistry letters vol. 13
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12.
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Ultrasensitive quantitative measurement of huntingtin phosphorylation at residue S13. [electronic resource] by
- Cariulo, Cristina
- Verani, Margherita
- Martufi, Paola
- Ingenito, Raffaele
- Finotto, Marco
- Deguire, Sean M
- Lavery, Daniel J
- Toledo-Sherman, Leticia
- Lee, Ramee
- Doherty, Elizabeth M
- Vogt, Thomas F
- Dominguez, Celia
- Lashuel, Hilal A
- Petricca, Lara
- Caricasole, Andrea
Producer: 20200727
In:
Biochemical and biophysical research communications vol. 521
Availability: No items available.
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13.
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2-Phenylamino-6-cyano-1H-benzimidazole-based isoform selective casein kinase 1 gamma (CK1γ) inhibitors. [electronic resource] by
- Hua, Zihao
- Huang, Xin
- Bregman, Howard
- Chakka, Nagasree
- DiMauro, Erin F
- Doherty, Elizabeth M
- Goldstein, Jon
- Gunaydin, Hakan
- Huang, Hongbing
- Mercede, Stephanie
- Newcomb, John
- Patel, Vinod F
- Turci, Susan M
- Yan, Jie
- Wilson, Cindy
- Martin, Matthew W
Producer: 20130107
In:
Bioorganic & medicinal chemistry letters vol. 22
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14.
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Discovery of pyridazinopyridinones as potent and selective p38 mitogen-activated protein kinase inhibitors. [electronic resource] by
- Wu, Bin
- Wang, Hui-Ling
- Pettus, Liping
- Wurz, Ryan P
- Doherty, Elizabeth M
- Henkle, Bradley
- McBride, Helen J
- Saris, Christiaan J M
- Wong, Lu Min
- Plant, Matthew H
- Sherman, Lisa
- Lee, Matthew R
- Hsieh, Faye
- Tasker, Andrew S
Producer: 20100930
In:
Journal of medicinal chemistry vol. 53
Availability: No items available.
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15.
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Novel vanilloid receptor-1 antagonists: 3. The identification of a second-generation clinical candidate with improved physicochemical and pharmacokinetic properties. [electronic resource] by
- Wang, Hui-Ling
- Katon, Jodie
- Balan, Chenera
- Bannon, Anthony W
- Bernard, Charles
- Doherty, Elizabeth M
- Dominguez, Celia
- Gavva, Narender R
- Gore, Vijay
- Ma, Vu
- Nishimura, Nobuko
- Surapaneni, Sekhar
- Tang, Phi
- Tamir, Rami
- Thiel, Oliver
- Treanor, James J S
- Norman, Mark H
Producer: 20071015
In:
Journal of medicinal chemistry vol. 50
Availability: No items available.
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16.
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Discovery of potent, orally available vanilloid receptor-1 antagonists. Structure-activity relationship of N-aryl cinnamides. [electronic resource] by
- Doherty, Elizabeth M
- Fotsch, Christopher
- Bo, Yunxin
- Chakrabarti, Partha P
- Chen, Ning
- Gavva, Narender
- Han, Nianhe
- Kelly, Michael G
- Kincaid, John
- Klionsky, Lana
- Liu, Qingyian
- Ognyanov, Vassil I
- Tamir, Rami
- Wang, Xianghong
- Zhu, Jiawang
- Norman, Mark H
- Treanor, James J S
Producer: 20050217
In:
Journal of medicinal chemistry vol. 48
Availability: No items available.
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17.
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AMG 9810 [(E)-3-(4-t-butylphenyl)-N-(2,3-dihydrobenzo[b][1,4] dioxin-6-yl)acrylamide], a novel vanilloid receptor 1 (TRPV1) antagonist with antihyperalgesic properties. [electronic resource] by
- Gavva, Narender R
- Tamir, Rami
- Qu, Yusheng
- Klionsky, Lana
- Zhang, T J
- Immke, David
- Wang, Judy
- Zhu, Dawn
- Vanderah, Todd W
- Porreca, Frank
- Doherty, Elizabeth M
- Norman, Mark H
- Wild, Kenneth D
- Bannon, Anthony W
- Louis, Jean-Claude
- Treanor, James J S
Producer: 20050519
In:
The Journal of pharmacology and experimental therapeutics vol. 313
Availability: No items available.
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18.
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Novel vanilloid receptor-1 antagonists: 1. Conformationally restricted analogues of trans-cinnamides. [electronic resource] by
- Norman, Mark H
- Zhu, Jiawang
- Fotsch, Christopher
- Bo, Yunxin
- Chen, Ning
- Chakrabarti, Partha
- Doherty, Elizabeth M
- Gavva, Narender R
- Nishimura, Nobuko
- Nixey, Thomas
- Ognyanov, Vassil I
- Rzasa, Robert M
- Stec, Markian
- Surapaneni, Sekhar
- Tamir, Rami
- Viswanadhan, Vellarkad N
- Treanor, James J S
Producer: 20071015
In:
Journal of medicinal chemistry vol. 50
Availability: No items available.
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19.
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Novel vanilloid receptor-1 antagonists: 2. Structure-activity relationships of 4-oxopyrimidines leading to the selection of a clinical candidate. [electronic resource] by
- Doherty, Elizabeth M
- Fotsch, Christopher
- Bannon, Anthony W
- Bo, Yunxin
- Chen, Ning
- Dominguez, Celia
- Falsey, James
- Gavva, Narender R
- Katon, Jodie
- Nixey, Thomas
- Ognyanov, Vassil I
- Pettus, Liping
- Rzasa, Robert M
- Stec, Markian
- Surapaneni, Sekhar
- Tamir, Rami
- Zhu, Jiawang
- Treanor, James J S
- Norman, Mark H
Producer: 20071015
In:
Journal of medicinal chemistry vol. 50
Availability: No items available.
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20.
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Selective inhibitors of the mutant B-Raf pathway: discovery of a potent and orally bioavailable aminoisoquinoline. [electronic resource] by
- Smith, Adrian L
- DeMorin, Frenel F
- Paras, Nick A
- Huang, Qi
- Petkus, Jeffrey K
- Doherty, Elizabeth M
- Nixey, Thomas
- Kim, Joseph L
- Whittington, Douglas A
- Epstein, Linda F
- Lee, Matthew R
- Rose, Mark J
- Babij, Carol
- Fernando, Manory
- Hess, Kristen
- Le, Quynh
- Beltran, Pedro
- Carnahan, Josette
Producer: 20091124
In:
Journal of medicinal chemistry vol. 52
Availability: No items available.
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