Discovery of potent, orally available vanilloid receptor-1 antagonists. Structure-activity relationship of N-aryl cinnamides. [electronic resource]
Producer: 20050217Description: 71-90 p. digitalISSN:- 0022-2623
- Administration, Oral
- Animals
- Biochemistry -- methods
- Biological Availability
- CHO Cells -- drug effects
- Calcium -- metabolism
- Capsaicin -- pharmacology
- Cinnamates -- chemistry
- Cricetinae
- Cricetulus
- Humans
- Hydrogen-Ion Concentration
- Inhibitory Concentration 50
- Ion Channels -- antagonists & inhibitors
- Male
- Rats
- Rats, Sprague-Dawley
- Recombinant Proteins -- drug effects
- Structure-Activity Relationship
- TRPV Cation Channels
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Publication Type: Journal Article
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