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Hyperphosphorylation of glucosyl C6 carbons and altered structure of glycogen in the neurodegenerative epilepsy Lafora disease. [electronic resource] by
- Nitschke, Felix
- Wang, Peixiang
- Schmieder, Peter
- Girard, Jean-Marie
- Awrey, Donald E
- Wang, Tony
- Israelian, Johan
- Zhao, XiaoChu
- Turnbull, Julie
- Heydenreich, Matthias
- Kleinpeter, Erich
- Steup, Martin
- Minassian, Berge A
Producer: 20140331
In:
Cell metabolism vol. 17
Availability: No items available.
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6.
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Spiro-naphthyridinone piperidines as inhibitors of S. aureus and E. coli enoyl-ACP reductase (FabI). [electronic resource] by
- Sampson, Peter B
- Picard, Christine
- Handerson, Sean
- McGrath, Teresa E
- Domagala, Megan
- Leeson, Andrew
- Romanov, Vladimir
- Awrey, Donald E
- Thambipillai, Dhushy
- Bardouniotis, Elias
- Kaplan, Nachum
- Berman, Judd M
- Pauls, Henry W
Producer: 20091123
In:
Bioorganic & medicinal chemistry letters vol. 19
Availability: No items available.
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7.
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Functional characterization of CFI-400945, a Polo-like kinase 4 inhibitor, as a potential anticancer agent. [electronic resource] by
- Mason, Jacqueline M
- Lin, Dan Chi-Chia
- Wei, Xin
- Che, Yi
- Yao, Yi
- Kiarash, Reza
- Cescon, David W
- Fletcher, Graham C
- Awrey, Donald E
- Bray, Mark R
- Pan, Guohua
- Mak, Tak W
Producer: 20141014
In:
Cancer cell vol. 26
Availability: No items available.
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8.
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2,3,4,5-Tetrahydro-1H-pyrido[2,3-b and e][1,4]diazepines as inhibitors of the bacterial enoyl ACP reductase, FabI. [electronic resource] by
- Ramnauth, Jailall
- Surman, Mathew D
- Sampson, Peter B
- Forrest, Bryan
- Wilson, Jeff
- Freeman, Emily
- Manning, David D
- Martin, Fernando
- Toro, Andras
- Domagala, Megan
- Awrey, Donald E
- Bardouniotis, Elias
- Kaplan, Nachum
- Berman, Judd
- Pauls, Henry W
Producer: 20091123
In:
Bioorganic & medicinal chemistry letters vol. 19
Availability: No items available.
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Design and optimization of (3-aryl-1H-indazol-6-yl)spiro[cyclopropane-1,3'-indolin]-2'-ones as potent PLK4 inhibitors with oral antitumor efficacy. [electronic resource] by
- Li, Sze-Wan
- Liu, Yong
- Sampson, Peter B
- Patel, Narendra Kumar
- Forrest, Bryan T
- Edwards, Louise
- Laufer, Radoslaw
- Feher, Miklos
- Ban, Fuqiang
- Awrey, Donald E
- Hodgson, Richard
- Beletskaya, Irina
- Mao, Guodong
- Mason, Jacqueline M
- Wei, Xin
- Luo, Xunyi
- Kiarash, Reza
- Green, Erin
- Mak, Tak W
- Pan, Guohua
- Pauls, Henry W
Producer: 20170815
In:
Bioorganic & medicinal chemistry letters vol. 26
Availability: No items available.
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10.
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The discovery of PLK4 inhibitors: (E)-3-((1H-Indazol-6-yl)methylene)indolin-2-ones as novel antiproliferative agents. [electronic resource] by
- Laufer, Radoslaw
- Forrest, Bryan
- Li, Sze-Wan
- Liu, Yong
- Sampson, Peter
- Edwards, Louise
- Lang, Yunhui
- Awrey, Donald E
- Mao, Guodong
- Plotnikova, Olga
- Leung, Genie
- Hodgson, Richard
- Beletskaya, Irina
- Mason, Jacqueline M
- Luo, Xunyi
- Wei, Xin
- Yao, Yi
- Feher, Miklos
- Ban, Fuqiang
- Kiarash, Reza
- Green, Erin
- Mak, Tak W
- Pan, Guohua
- Pauls, Henry W
Producer: 20131111
In:
Journal of medicinal chemistry vol. 56
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Discovery of 4-(4-aminopyrazolo[1,5-a][1,3,5]triazin-8-yl)benzamides as novel, highly potent and selective, orally bioavailable inhibitors of Tyrosine Threonine Kinase, TTK. [electronic resource] by
- Laufer, Radoslaw
- Li, Sze-Wan
- Liu, Yong
- Ng, Grace
- Lang, Yunhui
- Feher, Miklos
- Brokx, Richard
- Beletskaya, Irina
- Hodgson, Richard
- Mao, Guodong
- Plotnikova, Olga
- Awrey, Donald E
- Mason, Jacqueline M
- Wei, Xin
- Lin, Dan Chi-Chia
- Che, Yi
- Kiarash, Reza
- Madeira, Brian
- Fletcher, Graham C
- Mak, Tak W
- Bray, Mark R
- Pauls, Henry W
Producer: 20170619
In:
Bioorganic & medicinal chemistry letters vol. 26
Availability: No items available.
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12.
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The discovery of Polo-like kinase 4 inhibitors: identification of (1R,2S).2-(3-((E).4-(((cis).2,6-dimethylmorpholino)methyl)styryl). 1H.indazol-6-yl)-5'-methoxyspiro[cyclopropane-1,3'-indolin]-2'-one (CFI-400945) as a potent, orally active antitumor agent. [electronic resource] by
- Sampson, Peter B
- Liu, Yong
- Forrest, Bryan
- Cumming, Graham
- Li, Sze-Wan
- Patel, Narendra Kumar
- Edwards, Louise
- Laufer, Radoslaw
- Feher, Miklos
- Ban, Fuqiang
- Awrey, Donald E
- Mao, Guodong
- Plotnikova, Olga
- Hodgson, Richard
- Beletskaya, Irina
- Mason, Jacqueline M
- Luo, Xunyi
- Nadeem, Vincent
- Wei, Xin
- Kiarash, Reza
- Madeira, Brian
- Huang, Ping
- Mak, Tak W
- Pan, Guohua
- Pauls, Henry W
Producer: 20150427
In:
Journal of medicinal chemistry vol. 58
Availability: No items available.
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13.
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The discovery of Polo-like kinase 4 inhibitors: design and optimization of spiro[cyclopropane-1,3'[3H]indol]-2'(1'H).ones as orally bioavailable antitumor agents. [electronic resource] by
- Sampson, Peter B
- Liu, Yong
- Patel, Narendra Kumar
- Feher, Miklos
- Forrest, Bryan
- Li, Sze-Wan
- Edwards, Louise
- Laufer, Radoslaw
- Lang, Yunhui
- Ban, Fuqiang
- Awrey, Donald E
- Mao, Guodong
- Plotnikova, Olga
- Leung, Genie
- Hodgson, Richard
- Mason, Jacqueline M
- Wei, Xin
- Kiarash, Reza
- Green, Erin
- Qiu, Wei
- Chirgadze, Nickolay Y
- Mak, Tak W
- Pan, Guohua
- Pauls, Henry W
Producer: 20150427
In:
Journal of medicinal chemistry vol. 58
Availability: No items available.
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14.
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Discovery of Pyrazolo[1,5-a]pyrimidine TTK Inhibitors: CFI-402257 is a Potent, Selective, Bioavailable Anticancer Agent. [electronic resource] by
- Liu, Yong
- Laufer, Radoslaw
- Patel, Narendra Kumar
- Ng, Grace
- Sampson, Peter B
- Li, Sze-Wan
- Lang, Yunhui
- Feher, Miklos
- Brokx, Richard
- Beletskaya, Irina
- Hodgson, Richard
- Plotnikova, Olga
- Awrey, Donald E
- Qiu, Wei
- Chirgadze, Nickolay Y
- Mason, Jacqueline M
- Wei, Xin
- Lin, Dan Chi-Chia
- Che, Yi
- Kiarash, Reza
- Fletcher, Graham C
- Mak, Tak W
- Bray, Mark R
- Pauls, Henry W
Producer: 20160720
In:
ACS medicinal chemistry letters vol. 7
Availability: No items available.
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15.
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The Discovery of Orally Bioavailable Tyrosine Threonine Kinase (TTK) Inhibitors: 3-(4-(heterocyclyl)phenyl)-1H-indazole-5-carboxamides as Anticancer Agents. [electronic resource] by
- Liu, Yong
- Lang, Yunhui
- Patel, Narendra Kumar
- Ng, Grace
- Laufer, Radoslaw
- Li, Sze-Wan
- Edwards, Louise
- Forrest, Bryan
- Sampson, Peter B
- Feher, Miklos
- Ban, Fuqiang
- Awrey, Donald E
- Beletskaya, Irina
- Mao, Guodong
- Hodgson, Richard
- Plotnikova, Olga
- Qiu, Wei
- Chirgadze, Nickolay Y
- Mason, Jacqueline M
- Wei, Xin
- Lin, Dan Chi-Chia
- Che, Yi
- Kiarash, Reza
- Madeira, Brian
- Fletcher, Graham C
- Mak, Tak W
- Bray, Mark R
- Pauls, Henry W
Producer: 20150629
In:
Journal of medicinal chemistry vol. 58
Availability: No items available.
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