Results
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21.
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Optimization of Hydroxyethylamine Transition State Isosteres as Aspartic Protease Inhibitors by Exploiting Conformational Preferences. [electronic resource] by
- Bueno, Ana B
- Agejas, Javier
- Broughton, Howard
- Dally, Robert
- Durham, Timothy B
- Espinosa, Juan Félix
- González, Rosario
- Hahn, Patric J
- Marcos, Alicia
- Rodríguez, Ramón
- Sanz, Gema
- Soriano, José F
- Timm, David
- Vidal, Paloma
- Yang, Hsiu-Chiung
- McCarthy, James R
Producer: 20171229
In:
Journal of medicinal chemistry vol. 60
Availability: No items available.
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22.
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Potent, orally active corticotropin-releasing factor receptor-1 antagonists containing a tricyclic pyrrolopyridine or pyrazolopyridine core. [electronic resource] by
- Dyck, Brian
- Grigoriadis, Dimitri E
- Gross, Raymond S
- Guo, Zhiqiang
- Haddach, Mustapha
- Marinkovic, Dragan
- McCarthy, James R
- Moorjani, Manisha
- Regan, Collin F
- Saunders, John
- Schwaebe, Michael K
- Szabo, Tomas
- Williams, John P
- Zhang, Xiaohu
- Bozigian, Haig
- Chen, Ta Kung
Producer: 20050706
In:
Journal of medicinal chemistry vol. 48
Availability: No items available.
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23.
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Synthesis, crystallization, and biological evaluation of an orally active prodrug of gemcitabine. [electronic resource] by
- Bender, David M
- Bao, Jingqi
- Dantzig, Anne H
- Diseroad, William D
- Law, Kevin L
- Magnus, Nicholas A
- Peterson, Jeffrey A
- Perkins, Everett J
- Pu, Yangwei J
- Reutzel-Edens, Susan M
- Remick, David M
- Starling, James J
- Stephenson, Gregory A
- Vaid, Radhe K
- Zhang, Deyi
- McCarthy, James R
Producer: 20091221
In:
Journal of medicinal chemistry vol. 52
Availability: No items available.
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24.
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Biochemical and kinetic characterization of BACE1: investigation into the putative species-specificity for beta- and beta'-cleavage sites by human and murine BACE1. [electronic resource] by
- Yang, Hsiu-Chiung
- Chai, Xiyun
- Mosior, Marian
- Kohn, Wayne
- Boggs, Leonard N
- Erickson, Jon A
- McClure, Don B
- Yeh, Wu-Kuang
- Zhang, Lianshen
- Gonzalez-DeWhitt, Patricia
- Mayer, John P
- Martin, Jose Alfredo
- Hu, Jingdan
- Chen, Shu-Hui
- Bueno, Ana Belen
- Little, Sheila P
- McCarthy, James R
- May, Patrick C
Producer: 20050121
In:
Journal of neurochemistry vol. 91
Availability: No items available.
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25.
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Design and synthesis of tricyclic imidazo[4,5-b]pyridin-2-ones as corticotropin-releasing factor-1 antagonists. [electronic resource] by
- Guo, Zhiqiang
- Tellew, John E
- Gross, Raymond S
- Dyck, Brian
- Grey, Jonathan
- Haddach, Mustapha
- Kiankarimi, Mehrak
- Lanier, Marion
- Li, Bin-Feng
- Luo, Zhiyong
- McCarthy, James R
- Moorjani, Manisha
- Saunders, John
- Sullivan, Robert
- Zhang, Xiaohu
- Zamani-Kord, Said
- Grigoriadis, Dimitri E
- Crowe, Paul D
- Chen, Ta Kung
- Williams, John P
Producer: 20050927
In:
Journal of medicinal chemistry vol. 48
Availability: No items available.
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26.
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A tailored therapy for the metabolic syndrome: the dual peroxisome proliferator-activated receptor-alpha/gamma agonist LY465608 ameliorates insulin resistance and diabetic hyperglycemia while improving cardiovascular risk factors in preclinical models. [electronic resource] by
- Etgen, Garret J
- Oldham, Brian A
- Johnson, William T
- Broderick, Carol L
- Montrose, Chahrzad R
- Brozinick, Joseph T
- Misener, Elizabeth A
- Bean, James S
- Bensch, William R
- Brooks, Dawn A
- Shuker, Anthony J
- Rito, Christopher J
- McCarthy, James R
- Ardecky, Robert J
- Tyhonas, John S
- Dana, Sharon L
- Bilakovics, James M
- Paterniti, James R
- Ogilvie, Kathleen M
- Liu, Sha
- Kauffman, Raymond F
Producer: 20020510
In:
Diabetes vol. 51
Availability: No items available.
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27.
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Conversion of human-selective PPARalpha agonists to human/mouse dual agonists: a molecular modeling analysis. [electronic resource] by
- Wang, Minmin
- Winneroski, Leonard L
- Ardecky, Robert J
- Babine, Robert E
- Brooks, Dawn A
- Etgen, Garret J
- Hutchison, Darrell R
- Kauffman, Raymond F
- Kunkel, Aaron
- Mais, Dale E
- Montrose-Rafizadeh, Chahrzad
- Ogilvie, Kathleen M
- Oldham, Brian A
- Peters, Mary K
- Rito, Christopher J
- Rungta, Deepa K
- Tripp, Allie E
- Wilson, Sarah B
- Xu, Yanping
- Zink, Richard W
- McCarthy, James R
Producer: 20050420
In:
Bioorganic & medicinal chemistry letters vol. 14
Availability: No items available.
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28.
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Design and synthesis of alpha-aryloxy-alpha-methylhydrocinnamic acids: a novel class of dual peroxisome proliferator-activated receptor alpha/gamma agonists. [electronic resource] by
- Xu, Yanping
- Rito, Christopher J
- Etgen, Garret J
- Ardecky, Robert J
- Bean, James S
- Bensch, William R
- Bosley, Jacob R
- Broderick, Carol L
- Brooks, Dawn A
- Dominianni, Samuel J
- Hahn, Patric J
- Liu, Sha
- Mais, Dale E
- Montrose-Rafizadeh, Chahrzad
- Ogilvie, Kathy M
- Oldham, Brian A
- Peters, Mary
- Rungta, Deepa K
- Shuker, Anthony J
- Stephenson, Gregory A
- Tripp, Allie E
- Wilson, Sarah B
- Winneroski, Leonard L
- Zink, Richard
- Kauffman, Raymond F
- McCarthy, James R
Producer: 20040616
In:
Journal of medicinal chemistry vol. 47
Availability: No items available.
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