Design and synthesis of tricyclic imidazo[4,5-b]pyridin-2-ones as corticotropin-releasing factor-1 antagonists. [electronic resource]
Producer: 20050927Description: 5104-7 p. digitalISSN:- 0022-2623
- Administration, Oral
- Adrenocorticotropic Hormone -- blood
- Animals
- Blood-Brain Barrier -- metabolism
- CHO Cells
- Corticotropin-Releasing Hormone -- pharmacology
- Cricetinae
- Cricetulus
- Cyclic AMP -- antagonists & inhibitors
- Drug Design
- Heterocyclic Compounds, 3-Ring -- chemical synthesis
- Humans
- Imidazoles -- chemical synthesis
- Injections, Intravenous
- Male
- Pyridines -- chemical synthesis
- Radioligand Assay
- Rats
- Rats, Sprague-Dawley
- Receptors, Corticotropin-Releasing Hormone -- antagonists & inhibitors
- Stereoisomerism
- Structure-Activity Relationship
- CRF Receptor, Type 1
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Publication Type: Journal Article
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