Acquired resistance to IDH inhibition through trans or cis dimer-interface mutations. [electronic resource]
Producer: 20181211Description: 125-129 p. digitalISSN:- 1476-4687
- Alleles
- Allosteric Site -- drug effects
- Aminopyridines -- chemistry
- Animals
- Clinical Trials, Phase I as Topic
- Clinical Trials, Phase II as Topic
- Disease Progression
- Drug Resistance, Neoplasm -- drug effects
- Enzyme Inhibitors -- chemistry
- Female
- Glutamine -- genetics
- Glutarates -- blood
- HEK293 Cells
- Humans
- Isocitrate Dehydrogenase -- antagonists & inhibitors
- Isoleucine -- genetics
- Leukemia, Myeloid, Acute -- blood
- Mice
- Mice, Inbred C57BL
- Models, Molecular
- Mutant Proteins -- antagonists & inhibitors
- Mutation
- Protein Multimerization -- genetics
- Triazines -- chemistry
No physical items for this record
Publication Type: Case Reports; Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't
There are no comments on this title.
Log in to your account to post a comment.