Discovery and optimization of piperazine-1-thiourea-based human phosphoglycerate dehydrogenase inhibitors. (Record no. 28194815)
[ view plain ]
| 000 -LEADER | |
|---|---|
| fixed length control field | 01731 a2200481 4500 |
| 005 - DATE AND TIME OF LATEST TRANSACTION | |
| control field | 20250517205058.0 |
| 008 - FIXED-LENGTH DATA ELEMENTS--GENERAL INFORMATION | |
| fixed length control field | 201810s 0 0 eng d |
| 022 ## - INTERNATIONAL STANDARD SERIAL NUMBER | |
| International Standard Serial Number | 1464-3391 |
| 024 7# - OTHER STANDARD IDENTIFIER | |
| Standard number or code | 10.1016/j.bmc.2018.02.016 |
| Source of number or code | doi |
| 040 ## - CATALOGING SOURCE | |
| Original cataloging agency | NLM |
| Language of cataloging | eng |
| Transcribing agency | NLM |
| 100 1# - MAIN ENTRY--PERSONAL NAME | |
| Personal name | Rohde, Jason M |
| 264 #0 - PRODUCTION, PUBLICATION, DISTRIBUTION, MANUFACTURE, AND COPYRIGHT NOTICE | |
| Date of production, publication, distribution, manufacture, or copyright notice | 20181005 |
| 245 00 - TITLE STATEMENT | |
| Title | Discovery and optimization of piperazine-1-thiourea-based human phosphoglycerate dehydrogenase inhibitors. |
| Medium | [electronic resource] |
| 260 ## - PUBLICATION, DISTRIBUTION, ETC. | |
| Name of publisher, distributor, etc. | Bioorganic & medicinal chemistry |
| Date of publication, distribution, etc. | 05 2018 |
| 300 ## - PHYSICAL DESCRIPTION | |
| Extent | 1727-1739 p. |
| Other physical details | digital |
| 500 ## - GENERAL NOTE | |
| General note | Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't |
| 650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
| Topical term or geographic name entry element | Dose-Response Relationship, Drug |
| 650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
| Topical term or geographic name entry element | Drug Discovery |
| 650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
| Topical term or geographic name entry element | Enzyme Inhibitors |
| General subdivision | chemical synthesis |
| 650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
| Topical term or geographic name entry element | High-Throughput Screening Assays |
| 650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
| Topical term or geographic name entry element | Humans |
| 650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
| Topical term or geographic name entry element | Molecular Structure |
| 650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
| Topical term or geographic name entry element | Phosphoglycerate Dehydrogenase |
| General subdivision | antagonists & inhibitors |
| 650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
| Topical term or geographic name entry element | Piperazines |
| General subdivision | chemical synthesis |
| 650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
| Topical term or geographic name entry element | Structure-Activity Relationship |
| 650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
| Topical term or geographic name entry element | Thiourea |
| General subdivision | analogs & derivatives |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Brimacombe, Kyle R |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Liu, Li |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Pacold, Michael E |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Yasgar, Adam |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Cheff, Dorian M |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Lee, Tobie D |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Rai, Ganesha |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Baljinnyam, Bolormaa |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Li, Zhuyin |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Simeonov, Anton |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Hall, Matthew D |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Shen, Min |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Sabatini, David M |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Boxer, Matthew B |
| 773 0# - HOST ITEM ENTRY | |
| Title | Bioorganic & medicinal chemistry |
| Related parts | vol. 26 |
| -- | no. 8 |
| -- | p. 1727-1739 |
| 856 40 - ELECTRONIC LOCATION AND ACCESS | |
| Uniform Resource Identifier | <a href="https://doi.org/10.1016/j.bmc.2018.02.016">https://doi.org/10.1016/j.bmc.2018.02.016</a> |
| Public note | Available from publisher's website |
No items available.