Results
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Lack of protection with a novel, selective melanocortin receptor subtype-4 agonist RY767 in a rat transient middle cerebral artery occlusion stroke model. [electronic resource] by
- Regan, Christopher
- Shepherd, Cherrie
- Strack, Alison
- Weinberg, David
- Nargund, Ravi
- Ye, Zhixiong
- Pollard, Patrick
- Fong, Tung
- Reynolds, Ian
- Lynch, Joseph
Producer: 20090206
In:
Pharmacology vol. 83
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4.
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Development of a pharmaceutical cocrystal of a monophosphate salt with phosphoric acid. [electronic resource] by
- Chen, Alex M
- Ellison, Martha E
- Peresypkin, Andrey
- Wenslow, Robert M
- Variankaval, Narayan
- Savarin, Cecile G
- Natishan, Theresa K
- Mathre, David J
- Dormer, Peter G
- Euler, Danielle H
- Ball, Richard G
- Ye, Zhixiong
- Wang, Yaling
- Santos, Ivan
Producer: 20070326
In:
Chemical communications (Cambridge, England) no. 4
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5.
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Structure-activity relationship of linear tetrapeptides Tic-DPhe-Arg-Trp-NH2 at the human melanocortin-4 receptor and effects on feeding behaviors in rat. [electronic resource] by
- Ye, Zhixiong
- MacNeil, Tanya
- Weinberg, David H
- Kalyani, Rubana N
- Tang, Rui
- Strack, Alison M
- Murphy, Beth A
- Mosley, Ralph T
- Euan MacIntyre, D
- Van der Ploeg, Lex H T
- Patchett, Arthur A
- Wyvratt, Matthew J
- Nargund, Ravi P
Producer: 20080605
In:
Peptides vol. 26
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6.
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Melanocortin subtype 4 receptor agonists: structure-activity relationships about the 4-alkyl piperidine core. [electronic resource] by
- Sebhat, Iyassu K
- Lai, Yingjie
- Barakat, Khaled
- Ye, Zhixiong
- Tang, Rui
- Kalyani, Rubana N
- Vongs, Aurawan
- Macneil, Tanya
- Weinberg, David H
- Cabello, M Angeles
- Maroto, Marta
- Teran, Ana
- Fong, Tung M
- Van der Ploeg, Lex H T
- Patchett, Arthur A
- Nargund, Ravi P
Producer: 20071212
In:
Bioorganic & medicinal chemistry letters vol. 17
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7.
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Synthesis and SAR of potent and orally bioavailable tert-butylpyrrolidine archetype derived melanocortin subtype-4 receptor modulators. [electronic resource] by
- Guo, Liangqin
- Ye, Zhixiong
- Ujjainwalla, Feroze
- Sings, Heather L
- Sebhat, Iyassu K
- Huber, John
- Weinberg, David H
- Tang, Rui
- MacNeil, Tanya
- Tamvakopoulos, Constantin
- Peng, Qianping
- MacIntyre, Euan
- van der Ploeg, Lex H T
- Goulet, Mark T
- Wyvratt, Matthew J
- Nargund, Ravi P
Producer: 20080709
In:
Bioorganic & medicinal chemistry letters vol. 18
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8.
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Stimulation of Glucose-Dependent Insulin Secretion by a Potent, Selective sst3 Antagonist. [electronic resource] by
- Pasternak, Alexander
- Feng, Zhe
- de Jesus, Reynalda
- Ye, Zhixiong
- He, Shuwen
- Dobbelaar, Peter
- Bradley, Scott A
- Chicchi, Gary G
- Tsao, Kwei-Lan
- Trusca, Dorina
- Eiermann, George J
- Li, Cai
- Feng, Yue
- Wu, Margaret
- Shao, Qing
- Zhang, Bei B
- Nargund, Ravi
- Mills, Sander G
- Howard, Andrew D
- Yang, Lihu
- Zhou, Yun-Ping
Producer: 20140605
In:
ACS medicinal chemistry letters vol. 3
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9.
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1-Amino-1,2,3,4-tetrahydronaphthalene-2-carboxylic acid as a Tic mimetic: application in the synthesis of potent human melanocortin-4 receptor selective agonists. [electronic resource] by
- Bakshi, Raman K
- Hong, Qingmei
- Olson, J T
- Ye, Zhixiong
- Sebhat, Iyassue K
- Weinberg, David H
- MacNeil, Tanya
- Kalyani, Rubana N
- Tang, Rui
- Martin, William J
- Strack, Alison
- McGowan, Erin
- Tamvakopoulos, Constantin
- Miller, Randy R
- Stearns, Ralph A
- Tang, Wei
- Maclntyre, D Euan
- van der Ploeg, Lex H T
- Patchett, Arthur A
- Nargund, Ravi P
Producer: 20051219
In:
Bioorganic & medicinal chemistry letters vol. 15
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10.
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Discovery of potent, selective, and orally bioavailable 3H-spiro[isobenzofuran-1,4'-piperidine] based melanocortin subtype-4 receptor agonists. [electronic resource] by
- Guo, Liangqin
- Ye, Zhixiong
- Liu, Jian
- He, Shuwen
- Bakshi, Raman K
- Sebhat, Iyassu K
- Dobbelaar, Peter H
- Hong, Qingmei
- Jian, Tianying
- Dellureficio, James P
- Tsou, Nancy N
- Ball, Richard G
- Weinberg, David H
- MacNeil, Tanya
- Tang, Rui
- Tamvakopoulos, Constantin
- Peng, Qianping
- Chen, Howard Y
- Chen, Airu S
- Martin, William J
- MacIntyre, D Euan
- Strack, Alison M
- Fong, Tung M
- Wyvratt, Matthew J
- Nargund, Ravi P
Producer: 20101110
In:
Bioorganic & medicinal chemistry letters vol. 20
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11.
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Spiroindane based amides as potent and selective MC4R agonists for the treatment of obesity. [electronic resource] by
- He, Shuwen
- Ye, Zhixiong
- Dobbelaar, Peter H
- Sebhat, Iyassu K
- Guo, Liangqin
- Liu, Jian
- Jian, Tianying
- Lai, Yingjie
- Franklin, Christopher L
- Bakshi, Raman K
- Dellureficio, James P
- Hong, Qingmei
- Weinberg, David H
- Macneil, Tanya
- Tang, Rui
- Strack, Alison M
- Tamvakopoulos, Constantin
- Peng, Qianping
- Miller, Randy R
- Stearns, Ralph A
- Chen, Howard Y
- Chen, Airu S
- Fong, Tung M
- Wyvratt, Matthew J
- Nargund, Ravi P
Producer: 20101123
In:
Bioorganic & medicinal chemistry letters vol. 20
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12.
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Discovery of a piperazine urea based compound as a potent, selective, orally bioavailable melanocortin subtype-4 receptor partial agonist. [electronic resource] by
- Hong, Qingmei
- Bakshi, Raman K
- Palucki, Brenda L
- Park, Min K
- Ye, Zhixiong
- He, Shuwen
- Pollard, Patrick G
- Sebhat, Iyassu K
- Liu, Jian
- Guo, Liangqin
- Cashen, Doreen E
- Martin, William J
- Weinberg, David H
- MacNeil, Tanya
- Tang, Rui
- Tamvakopoulos, Constantin
- Peng, Qianping
- Miller, Randy R
- Stearns, Ralph A
- Chen, Howard Y
- Chen, Airu S
- Strack, Alison M
- Fong, Tung M
- MacIntyre, D Euan
- Wyvratt, Matthew J
- Nargund, Ravi P
Producer: 20110719
In:
Bioorganic & medicinal chemistry letters vol. 21
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13.
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Discovery of highly potent and efficacious MC4R agonists with spiroindane N-Me-1,2,4-triazole privileged structures for the treatment of obesity. [electronic resource] by
- He, Shuwen
- Ye, Zhixiong
- Dobbelaar, Peter H
- Bakshi, Raman K
- Hong, Qingmei
- Dellureficio, James P
- Sebhat, Iyassu K
- Guo, Liangqin
- Liu, Jian
- Jian, Tianying
- Lai, Yingjie
- Franklin, Christopher L
- Reibarkh, Mikhail
- Holmes, Mark A
- Weinberg, David H
- MacNeil, Tanya
- Tang, Rui
- Tamvakopoulos, Constantin
- Peng, Qianping
- Miller, Randy R
- Stearns, Ralph A
- Chen, Howard Y
- Chen, Airu S
- Strack, Alison M
- Fong, Tung M
- Wyvratt, Matthew J
- Nargund, Ravi P
Producer: 20110329
In:
Bioorganic & medicinal chemistry letters vol. 20
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14.
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Design and pharmacology of N-[(3R)-1,2,3,4-tetrahydroisoquinolinium- 3-ylcarbonyl]-(1R)-1-(4-chlorobenzyl)- 2-[4-cyclohexyl-4-(1H-1,2,4-triazol- 1-ylmethyl)piperidin-1-yl]-2-oxoethylamine (1), a potent, selective, melanocortin subtype-4 receptor agonist. [electronic resource] by
- Sebhat, Iyassu K
- Martin, William J
- Ye, Zhixiong
- Barakat, Khaled
- Mosley, Ralph T
- Johnston, David B R
- Bakshi, Raman
- Palucki, Brenda
- Weinberg, David H
- MacNeil, Tanya
- Kalyani, Rubana N
- Tang, Rui
- Stearns, Ralph A
- Miller, Randy R
- Tamvakopoulos, Constantin
- Strack, Alison M
- McGowan, Erin
- Cashen, Doreen E
- Drisko, Jennifer E
- Hom, Gary J
- Howard, Andrew D
- MacIntyre, D Euan
- van der Ploeg, Lex H T
- Patchett, Arthur A
- Nargund, Ravi P
Producer: 20021105
In:
Journal of medicinal chemistry vol. 45
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15.
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Discovery of (2S)-N-[(1R)-2-[4-cyclohexyl-4-[[(1,1-dimethylethyl)amino]carbonyl]-1-piperidinyl]-1-[(4-fluorophenyl)methyl]-2-oxoethyl]-4-methyl-2-piperazinecarboxamide (MB243), a potent and selective melanocortin subtype-4 receptor agonist. [electronic resource] by
- Palucki, Brenda L
- Park, Min K
- Nargund, Ravi P
- Ye, Zhixiong
- Sebhat, Iyassu K
- Pollard, Patrick G
- Kalyani, Rubana N
- Tang, Rui
- Macneil, Tanya
- Weinberg, David H
- Vongs, Aurawan
- Rosenblum, Charles I
- Doss, George A
- Miller, Randall R
- Stearns, Ralph A
- Peng, Qianping
- Tamvakopoulos, Constantin
- McGowan, Erin
- Martin, William J
- Metzger, Joseph M
- Shepherd, Cherrie A
- Strack, Alison M
- Macintyre, D Euan
- Van der Ploeg, Lex H T
- Patchett, Arthur A
Producer: 20050502
In:
Bioorganic & medicinal chemistry letters vol. 15
Availability: No items available.
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16.
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Discovery of a spiroindane based compound as a potent, selective, orally bioavailable melanocortin subtype-4 receptor agonist. [electronic resource] by
- He, Shuwen
- Ye, Zhixiong
- Dobbelaar, Peter H
- Sebhat, Iyassu K
- Guo, Liangqin
- Liu, Jian
- Jian, Tianying
- Lai, Yingjie
- Franklin, Christopher L
- Bakshi, Raman K
- Dellureficio, James P
- Hong, Qingmei
- Tsou, Nancy N
- Ball, Richard G
- Cashen, Doreen E
- Martin, William J
- Weinberg, David H
- Macneil, Tanya
- Tang, Rui
- Tamvakopoulos, Constantin
- Peng, Qianping
- Miller, Randy R
- Stearns, Ralph A
- Chen, Howard Y
- Chen, Airu S
- Strack, Alison M
- Fong, Tung M
- Macintyre, D Euan
- Wyvratt, Matthew J
- Nargund, Ravi P
Producer: 20100705
In:
Bioorganic & medicinal chemistry letters vol. 20
Availability: No items available.
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17.
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Discovery and activity of (1R,4S,6R)-N-[(1R)-2-[4-cyclohexyl-4-[[(1,1-dimethylethyl)amino]carbonyl]-1-piperidinyl]-1-[(4-fluorophenyl)methyl]-2-oxoethyl]-2-methyl-2-azabicyclo[2.2.2]octane-6-carboxamide (3, RY764), a potent and selective melanocortin subtype-4 receptor agonist. [electronic resource] by
- Ye, Zhixiong
- Guo, Liangqin
- Barakat, Khaled J
- Pollard, Patrick G
- Palucki, Brenda L
- Sebhat, Iyassu K
- Bakshi, Raman K
- Tang, Rui
- Kalyani, Rubana N
- Vongs, Aurawan
- Chen, Airu S
- Chen, Howard Y
- Rosenblum, Charles I
- MacNeil, Tanya
- Weinberg, David H
- Peng, Qianping
- Tamvakopoulos, Constantin
- Miller, Randy R
- Stearns, Ralph A
- Cashen, Doreen E
- Martin, William J
- Metzger, Joseph M
- Strack, Alison M
- MacIntyre, D Euan
- Van der Ploeg, Lex H T
- Patchett, Arthur A
- Wyvratt, Matthew J
- Nargund, Ravi P
Producer: 20051011
In:
Bioorganic & medicinal chemistry letters vol. 15
Availability: No items available.
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18.
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Optimization of privileged structures for selective and potent melanocortin subtype-4 receptor ligands. [electronic resource] by
- Hong, Qingmei
- Bakshi, Raman K
- Dellureficio, James
- He, Shuwen
- Ye, Zhixiong
- Dobbelaar, Peter H
- Sebhat, Iyassu K
- Guo, Liangqin
- Liu, Jian
- Jian, Tianying
- Tang, Rui
- Kalyani, Rubana N
- Macneil, Tanya
- Vongs, Aurawan
- Rosenblum, Charles I
- Weinberg, David H
- Peng, Qingping
- Tamvakopoulos, Constantin
- Miller, Randy R
- Stearns, Ralph A
- Cashen, Doreen
- Martin, Willian J
- Chen, Airu S
- Metzger, Joseph M
- Chen, Howard Y
- Strack, Allison M
- Fong, Tung M
- Maclntyre, Euan
- Van der Ploeg, Lex H T
- Wyvratt, Matthew J
- Nargund, Ravi P
Producer: 20101123
In:
Bioorganic & medicinal chemistry letters vol. 20
Availability: No items available.
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Investigation of Cardiovascular Effects of Tetrahydro-β-carboline sstr3 antagonists. [electronic resource] by
- He, Shuwen
- Lai, Zhong
- Ye, Zhixiong
- Dobbelaar, Peter H
- Shah, Shrenik K
- Truong, Quang
- Du, Wu
- Guo, Liangqin
- Liu, Jian
- Jian, Tianying
- Qi, Hongbo
- Bakshi, Raman K
- Hong, Qingmei
- Dellureficio, James
- Reibarkh, Mikhail
- Samuel, Koppara
- Reddy, Vijay B
- Mitelman, Stan
- Tong, Sharon X
- Chicchi, Gary G
- Tsao, Kwei-Lan
- Trusca, Dorina
- Wu, Margaret
- Shao, Qing
- Trujillo, Maria E
- Fernandez, Guillermo
- Nelson, Donald
- Bunting, Patricia
- Kerr, Janet
- Fitzgerald, Patrick
- Morissette, Pierre
- Volksdorf, Sylvia
- Eiermann, George J
- Li, Cai
- Zhang, Bei
- Howard, Andrew D
- Zhou, Yun-Ping
- Nargund, Ravi P
- Hagmann, William K
Producer: 20140722
In:
ACS medicinal chemistry letters vol. 5
Availability: No items available.
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20.
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The Discovery of MK-4256, a Potent SSTR3 Antagonist as a Potential Treatment of Type 2 Diabetes. [electronic resource] by
- He, Shuwen
- Ye, Zhixiong
- Truong, Quang
- Shah, Shrenik
- Du, Wu
- Guo, Liangqin
- Dobbelaar, Peter H
- Lai, Zhong
- Liu, Jian
- Jian, Tianying
- Qi, Hongbo
- Bakshi, Raman K
- Hong, Qingmei
- Dellureficio, James
- Pasternak, Alexander
- Feng, Zhe
- deJesus, Reynalda
- Yang, Lihu
- Reibarkh, Mikhail
- Bradley, Scott A
- Holmes, Mark A
- Ball, Richard G
- Ruck, Rebecca T
- Huffman, Mark A
- Wong, Frederick
- Samuel, Koppara
- Reddy, Vijay B
- Mitelman, Stan
- Tong, Sharon X
- Chicchi, Gary G
- Tsao, Kwei-Lan
- Trusca, Dorina
- Wu, Margaret
- Shao, Qing
- Trujillo, Maria E
- Eiermann, George J
- Li, Cai
- Zhang, Bei B
- Howard, Andrew D
- Zhou, Yun-Ping
- Nargund, Ravi P
- Hagmann, William K
Producer: 20140605
In:
ACS medicinal chemistry letters vol. 3
Availability: No items available.
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