In vitro phase I cytochrome P450 metabolism, permeability and pharmacokinetics of SB639, a novel histone deacetylase inhibitor in preclinical species. [electronic resource]
Producer: 20070627Description: 1021-4 p. digitalISSN:- 0918-6158
- Administration, Oral
- Animals
- Benzimidazoles -- blood
- Biological Availability
- Caco-2 Cells
- Cell Membrane Permeability -- drug effects
- Cytochrome P-450 Enzyme System -- metabolism
- Dogs
- Drug Evaluation, Preclinical
- Enzyme Inhibitors -- blood
- Female
- Half-Life
- Histone Deacetylase Inhibitors
- Humans
- Hydroxamic Acids -- blood
- Male
- Metabolic Detoxication, Phase I
- Mice
- Mice, Inbred BALB C
- Microsomes, Liver -- drug effects
- Pyrroles -- blood
- Pyrrolidines
- Rats
- Rats, Wistar
- Vorinostat
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Publication Type: Journal Article
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