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Pyrazoles as non-classical bioisosteres in prolylcarboxypeptidase (PrCP) inhibitors. [electronic resource] by
- Graham, Thomas H
- Shu, Min
- Verras, Andreas
- Chen, Qing
- Garcia-Calvo, Margarita
- Li, Xiaohua
- Lisnock, JeanMarie
- Tong, Xinchun
- Tung, Elaine C
- Wiltsie, Judyann
- Hale, Jeffrey J
- Pinto, Shirly
- Shen, Dong-Ming
Producer: 20150330
In:
Bioorganic & medicinal chemistry letters vol. 24
Availability: No items available.
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Evidence for the bioactivation of zomepirac and tolmetin by an oxidative pathway: identification of glutathione adducts in vitro in human liver microsomes and in vivo in rats. [electronic resource] by
- Chen, Qing
- Doss, George A
- Tung, Elaine C
- Liu, Wensheng
- Tang, Yui S
- Braun, Matthew P
- Didolkar, Varsha
- Strauss, John R
- Wang, Regina W
- Stearns, Ralph A
- Evans, David C
- Baillie, Thomas A
- Tang, Wei
Producer: 20060227
In:
Drug metabolism and disposition: the biological fate of chemicals vol. 34
Availability: No items available.
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6.
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Discovery of indazole aldosterone synthase (CYP11B2) inhibitors as potential treatments for hypertension. [electronic resource] by
- Hoyt, Scott B
- Taylor, Jerry
- London, Clare
- Ali, Amjad
- Ujjainwalla, Feroze
- Tata, Jim
- Struthers, Mary
- Cully, Doris
- Wisniewski, Tom
- Ren, Ning
- Bopp, Charlene
- Sok, Andrea
- Verras, Andreas
- McMasters, Daniel
- Chen, Qing
- Tung, Elaine
- Tang, Wei
- Salituro, Gino
- Clemas, Joe
- Zhou, Gaochao
- MacNeil, Douglas
- Duffy, Ruth
- Xiong, Yusheng
Producer: 20171219
In:
Bioorganic & medicinal chemistry letters vol. 27
Availability: No items available.
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Biochemical characterization of cholesteryl ester transfer protein inhibitors. [electronic resource] by
- Ranalletta, Mollie
- Bierilo, Kathleen K
- Chen, Ying
- Milot, Denise
- Chen, Qing
- Tung, Elaine
- Houde, Caroline
- Elowe, Nadine H
- Garcia-Calvo, Margarita
- Porter, Gene
- Eveland, Suzanne
- Frantz-Wattley, Betsy
- Kavana, Mike
- Addona, George
- Sinclair, Peter
- Sparrow, Carl
- O'Neill, Edward A
- Koblan, Ken S
- Sitlani, Ayesha
- Hubbard, Brian
- Fisher, Timothy S
Producer: 20110214
In:
Journal of lipid research vol. 51
Availability: No items available.
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8.
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A new class of prolylcarboxypeptidase inhibitors, part 2: the aminocyclopentanes. [electronic resource] by
- Graham, Thomas H
- Liu, Wensheng
- Verras, Andreas
- Reibarkh, Mikhail
- Bleasby, Kelly
- Bhatt, Urmi R
- Chen, Qing
- Garcia-Calvo, Margarita
- Geissler, Wayne M
- Gorski, Judith N
- He, Huaibing
- Lassman, Michael E
- Lisnock, JeanMarie
- Li, Xiaohua
- Shen, Zhu
- Tong, Xinchun
- Tung, Elaine C
- Wiltsie, Judyann
- Xie, Dan
- Xu, Suoyu
- Xiao, Jianying
- Hale, Jeffrey J
- Pinto, Shirly
- Shen, Dong-Ming
Producer: 20120918
In:
Bioorganic & medicinal chemistry letters vol. 22
Availability: No items available.
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Discovery and optimization of orally active cyclohexane-based prolylcarboxypeptidase (PrCP) inhibitors. [electronic resource] by
- Debenham, John S
- Graham, Thomas H
- Verras, Andreas
- Zhang, Yong
- Clements, Matthew J
- Kuethe, Jeffrey T
- Madsen-Duggan, Christina
- Liu, Wensheng
- Bhatt, Urmi R
- Chen, Dunlu
- Chen, Qing
- Garcia-Calvo, Margarita
- Geissler, Wayne M
- He, Huaibing
- Li, Xiaohua
- Lisnock, JeanMarie
- Shen, Zhu
- Tong, Xinchun
- Tung, Elaine C
- Wiltsie, Judyann
- Xu, Suoyu
- Hale, Jeffrey J
- Pinto, Shirly
- Shen, Dong-Ming
Producer: 20140817
In:
Bioorganic & medicinal chemistry letters vol. 23
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10.
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Discovery of Spirocyclic Aldosterone Synthase Inhibitors as Potential Treatments for Resistant Hypertension. [electronic resource] by
- Petrilli, Whitney L
- Hoyt, Scott B
- London, Clare
- McMasters, Daniel
- Verras, Andreas
- Struthers, Mary
- Cully, Doris
- Wisniewski, Thomas
- Ren, Ning
- Bopp, Charlene
- Sok, Andrea
- Chen, Qing
- Li, Ying
- Tung, Elaine
- Tang, Wei
- Salituro, Gino
- Knemeyer, Ian
- Karanam, Bindhu
- Clemas, Joseph
- Zhou, Gaochao
- Gibson, Jack
- Shipley, Carrie Ann
- MacNeil, Douglas J
- Duffy, Ruth
- Tata, James R
- Ujjainwalla, Feroze
- Ali, Amjad
- Xiong, Yusheng
Publication details: ACS medicinal chemistry letters Jan 2017
In:
ACS medicinal chemistry letters vol. 8
Availability: No items available.
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11.
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The discovery of non-benzimidazole and brain-penetrant prolylcarboxypeptidase inhibitors. [electronic resource] by
- Graham, Thomas H
- Shen, Hong C
- Liu, Wensheng
- Xiong, Yusheng
- Verras, Andreas
- Bleasby, Kelly
- Bhatt, Urmi R
- Chabin, Renee M
- Chen, Dunlu
- Chen, Qing
- Garcia-Calvo, Margarita
- Geissler, Wayne M
- He, Huaibing
- Lassman, Michael E
- Shen, Zhu
- Tong, Xinchun
- Tung, Elaine C
- Xie, Dan
- Xu, Suoyu
- Colletti, Steven L
- Tata, James R
- Hale, Jeffrey J
- Pinto, Shirly
- Shen, Dong-Ming
Producer: 20120803
In:
Bioorganic & medicinal chemistry letters vol. 22
Availability: No items available.
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12.
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A new class of prolylcarboxypeptidase inhibitors, part 1: discovery and evaluation. [electronic resource] by
- Graham, Thomas H
- Liu, Wensheng
- Verras, Andreas
- Sebhat, Iyassu K
- Xiong, Yusheng
- Bleasby, Kelly
- Bhatt, Urmi R
- Chen, Qing
- Garcia-Calvo, Margarita
- Geissler, Wayne M
- Gorski, Judith N
- He, Huaibing
- Lassman, Michael E
- Lisnock, JeanMarie
- Li, Xiaohua
- Shen, Zhu
- Tong, Xinchun
- Tung, Elaine C
- Wiltsie, Judyann
- Xiao, Jianying
- Xie, Dan
- Xu, Suoyu
- Hale, Jeffrey J
- Pinto, Shirly
- Shen, Dong-Ming
Producer: 20120918
In:
Bioorganic & medicinal chemistry letters vol. 22
Availability: No items available.
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13.
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Discovery of Triazole CYP11B2 Inhibitors with in Vivo Activity in Rhesus Monkeys. [electronic resource] by
- Hoyt, Scott B
- Petrilli, Whitney
- London, Clare
- Liang, Gui-Bai
- Tata, Jim
- Hu, Qingzhong
- Yin, Lina
- van Koppen, Chris J
- Hartmann, Rolf W
- Struthers, Mary
- Wisniewski, Tom
- Ren, Ning
- Bopp, Charlene
- Sok, Andrea
- Cai, Tian-Quan
- Stribling, Sloan
- Pai, Lee-Yuh
- Ma, Xiuying
- Metzger, Joe
- Verras, Andreas
- McMasters, Daniel
- Chen, Qing
- Tung, Elaine
- Tang, Wei
- Salituro, Gino
- Buist, Nicole
- Clemas, Joe
- Zhou, Gaochao
- Gibson, Jack
- Maxwell, Carrie Ann
- Lassman, Mike
- McLaughlin, Theresa
- Castro-Perez, Jose
- Szeto, Daphne
- Forrest, Gail
- Hajdu, Richard
- Rosenbach, Mark
- Xiong, Yusheng
Producer: 20150820
In:
ACS medicinal chemistry letters vol. 6
Availability: No items available.
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14.
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Discovery of Benzimidazole CYP11B2 Inhibitors with in Vivo Activity in Rhesus Monkeys. [electronic resource] by
- Hoyt, Scott B
- Park, Min K
- London, Clare
- Xiong, Yusheng
- Tata, Jim
- Bennett, D Jonathan
- Cooke, Andrew
- Cai, Jiaqiang
- Carswell, Emma
- Robinson, John
- MacLean, John
- Brown, Lindsay
- Belshaw, Simone
- Clarkson, Thomas R
- Liu, Kun
- Liang, Gui-Bai
- Struthers, Mary
- Cully, Doris
- Wisniewski, Tom
- Ren, Ning
- Bopp, Charlene
- Sok, Andrea
- Cai, Tian-Quan
- Stribling, Sloan
- Pai, Lee-Yuh
- Ma, Xiuying
- Metzger, Joe
- Verras, Andreas
- McMasters, Daniel
- Chen, Qing
- Tung, Elaine
- Tang, Wei
- Salituro, Gino
- Buist, Nicole
- Kuethe, Jeff
- Rivera, Nelo
- Clemas, Joe
- Zhou, Gaochao
- Gibson, Jack
- Maxwell, Carrie Ann
- Lassman, Mike
- McLaughlin, Theresa
- Castro-Perez, Jose
- Szeto, Daphne
- Forrest, Gail
- Hajdu, Richard
- Rosenbach, Mark
- Ali, Amjad
Producer: 20150525
In:
ACS medicinal chemistry letters vol. 6
Availability: No items available.
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