Design, Synthesis, and Biological Evaluation of Novel DNA Gyrase-Inhibiting Spiropyrimidinetriones as Potent Antibiotics for Treatment of Infections Caused by Multidrug-Resistant Gram-Positive Bacteria. [electronic resource]
Producer: 20200303Description: 2950-2973 p. digitalISSN:- 1520-4804
- Animals
- Anti-Bacterial Agents -- chemistry
- DNA Gyrase -- drug effects
- Dogs
- Drug Design
- Drug Resistance, Multiple, Bacterial -- drug effects
- Gram-Positive Bacteria -- drug effects
- Gram-Positive Bacterial Infections -- drug therapy
- Humans
- Mice
- Microbial Sensitivity Tests
- Rats
- Spiro Compounds -- chemistry
- Structure-Activity Relationship
- Topoisomerase II Inhibitors -- chemistry
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Publication Type: Journal Article; Research Support, Non-U.S. Gov't
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