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Hydroxyethylamine isostere of an HIV-1 protease inhibitor prefers its amine to the hydroxy group in binding to catalytic aspartates. A synchrotron study of HIV-1 protease in complex with a peptidomimetic inhibitor. [electronic resource] by
- Dohnálek, Jan
- Hasek, Jindrich
- Dusková, Jarmila
- Petroková, Hana
- Hradilek, Martin
- Soucek, Milan
- Konvalinka, Jan
- Brynda, Jirí
- Sedlácek, Juraj
- Fábry, Milan
Producer: 20020429
In:
Journal of medicinal chemistry vol. 45
Availability: No items available.
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8.
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A phenylnorstatine inhibitor binding to HIV-1 protease: geometry, protonation, and subsite-pocket interactions analyzed at atomic resolution. [electronic resource] by
- Brynda, Jiri
- Rezacova, Pavlina
- Fabry, Milan
- Horejsi, Magdalena
- Stouracova, Renata
- Sedlacek, Juraj
- Soucek, Milan
- Hradilek, Martin
- Lepsik, Martin
- Konvalinka, Jan
Producer: 20040519
In:
Journal of medicinal chemistry vol. 47
Availability: No items available.
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9.
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Stabilization of antibody structure upon association to a human carbonic anhydrase IX epitope studied by X-ray crystallography, microcalorimetry, and molecular dynamics simulations. [electronic resource] by
- Král, Vlastimil
- Mader, Pavel
- Collard, Renata
- Fábry, Milan
- Horejsí, Magdaléna
- Rezácová, Pavlína
- Kozísek, Milan
- Závada, Jan
- Sedlácek, Juraj
- Rulísek, Lubomír
- Brynda, Jirí
Producer: 20080815
In:
Proteins vol. 71
Availability: No items available.
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Role of hydroxyl group and R/S configuration of isostere in binding properties of HIV-1 protease inhibitors. [electronic resource] by
- Petroková, Hana
- Dusková, Jarmila
- Dohnálek, Jan
- Skálová, Tereza
- Vondrácková-Buchtelová, Eva
- Soucek, Milan
- Konvalinka, Jan
- Brynda, Jirí
- Fábry, Milan
- Sedlácek, Juraj
- Hasek, Jindrich
Producer: 20050303
In:
European journal of biochemistry vol. 271
Availability: No items available.
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11.
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Potent inhibition of drug-resistant HIV protease variants by monoclonal antibodies. [electronic resource] by
- Bartonová, Vanda
- Král, Vlastimil
- Sieglová, Irena
- Brynda, Jirí
- Fábry, Milan
- Horejsí, Magdalena
- Kozísek, Milan
- Sasková, Klára Grantz
- Konvalinka, Jan
- Sedlácek, Juraj
- Rezácová, Pavlína
Producer: 20080715
In:
Antiviral research vol. 78
Availability: No items available.
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12.
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On the role of the R configuration of the reaction-intermediate isostere in HIV-1 protease-inhibitor binding: X-ray structure at 2.0 A resolution. [electronic resource] by
- Dusková, Jarmila
- Dohnálek, Jan
- Skálová, Tereza
- Petroková, Hana
- Vondrácková, Eva
- Hradílek, Martin
- Konvalinka, Jan
- Soucek, Milan
- Brynda, Jirí
- Fábry, Milan
- Sedlácek, Juraj
- Hasek, Jindrich
Producer: 20060705
In:
Acta crystallographica. Section D, Biological crystallography vol. 62
Availability: No items available.
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13.
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From nonpeptide toward noncarbon protease inhibitors: metallacarboranes as specific and potent inhibitors of HIV protease. [electronic resource] by
- Cígler, Petr
- Kozísek, Milan
- Rezácová, Pavlína
- Brynda, Jírí
- Otwinowski, Zbyszek
- Pokorná, Jana
- Plesek, Jaromír
- Grüner, Bohumír
- Dolecková-Maresová, Lucie
- Mása, Martin
- Sedlácek, Juraj
- Bodem, Jochen
- Kräusslich, Hans-Georg
- Král, Vladimír
- Konvalinka, Jan
Producer: 20051212
In:
Proceedings of the National Academy of Sciences of the United States of America vol. 102
Availability: No items available.
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14.
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Design of HIV protease inhibitors based on inorganic polyhedral metallacarboranes. [electronic resource] by
- Rezácová, Pavlína
- Pokorná, Jana
- Brynda, Jirí
- Kozísek, Milan
- Cígler, Petr
- Lepsík, Martin
- Fanfrlík, Jindrich
- Rezác, Jan
- Grantz Sasková, Klára
- Sieglová, Irena
- Plesek, Jaromír
- Sícha, Václav
- Grüner, Bohumír
- Oberwinkler, Heike
- Sedlácek', Juraj
- Kräusslich, Hans-Georg
- Hobza, Pavel
- Král, Vladimír
- Konvalinka, Jan
Producer: 20091221
In:
Journal of medicinal chemistry vol. 52
Availability: No items available.
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