Fluoxetine- and norfluoxetine-mediated complex drug-drug interactions: in vitro to in vivo correlation of effects on CYP2D6, CYP2C19, and CYP3A4. [electronic resource]
Producer: 20140703Description: 653-62 p. digitalISSN:- 1532-6535
- Adult
- Antidepressive Agents, Second-Generation -- administration & dosage
- Area Under Curve
- Aryl Hydrocarbon Hydroxylases -- antagonists & inhibitors
- Biotransformation
- Computer Simulation
- Cytochrome P-450 CYP2C19
- Cytochrome P-450 CYP2D6 -- metabolism
- Cytochrome P-450 CYP2D6 Inhibitors
- Cytochrome P-450 CYP3A -- metabolism
- Cytochrome P-450 CYP3A Inhibitors
- Dextromethorphan -- pharmacokinetics
- Drug Interactions
- Female
- Fluoxetine -- administration & dosage
- Half-Life
- Hepatocytes -- drug effects
- Humans
- Lovastatin -- pharmacokinetics
- Male
- Midazolam -- pharmacokinetics
- Models, Statistical
- Omeprazole -- pharmacokinetics
- Stereoisomerism
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Publication Type: Journal Article; Research Support, N.I.H., Extramural
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