Results
|
1.
|
Synthesis of novel HIV protease inhibitors (PI) with activity against PI-resistant virus. [electronic resource] by
- Raghavan, Subharekha
- Lu, Zhijian
- Beeson, Teresa
- Chapman, Kevin T
- Schleif, William A
- Olsen, David B
- Stahlhut, Mark
- Rutkowski, Carrie A
- Gabryelski, Lori
- Emini, Emilio
- Tata, James R
Producer: 20071127
In:
Bioorganic & medicinal chemistry letters vol. 17
Availability: No items available.
|
|
2.
|
Selective Formation of Functionalized α-Quaternary Malononitriles toward 5,5-Disubstituted Pyrrolopyrimidinones. [electronic resource] by
- Whitehead, Alan
- Zhang, Yong
- McCabe Dunn, Jamie
- Sherer, Edward C
- Lam, Yu-Hong
- Stelmach, John
- Sun, Aaron
- Shiroda, Melisa
- Orr, Robert K
- Waddell, Sherman T
- Raghavan, Subharekha
Producer: 20180613
In:
Organic letters vol. 19
Availability: No items available.
|
|
3.
|
Combinatorial library of indinavir analogues: replacement for the aminoindanol at P2'. [electronic resource] by
- Raghavan, Subharekha
- Yang, Zheng
- Mosley, Ralph T
- Schleif, William A
- Gabryelski, Lori
- Olsen, David B
- Stahlhut, Mark
- Kuo, Lawrence C
- Emini, Emilio A
- Chapman, Kevin T
- Tata, James R
Producer: 20030311
In:
Bioorganic & medicinal chemistry letters vol. 12
Availability: No items available.
|
|
4.
|
The discovery of high affinity agonists of GPR109a with reduced serum shift and improved ADME properties. [electronic resource] by
- Imbriglio, Jason E
- DiRocco, Daniel
- Bodner, Rena
- Raghavan, Subharekha
- Chen, Weichun
- Marley, Daria
- Esser, Craig
- Holt, Tom G
- Wolff, Michael S
- Taggart, Andrew K P
- Waters, M Gerard
- Tata, James R
- Colletti, Steven L
Producer: 20110815
In:
Bioorganic & medicinal chemistry letters vol. 21
Availability: No items available.
|
|
5.
|
Design and synthesis of highly potent HIV protease inhibitors with activity against resistant virus. [electronic resource] by
- Lu, Zhijian
- Raghavan, Subharekha
- Bohn, Joann
- Charest, Mark
- Stahlhut, Mark W
- Rutkowski, Carrie A
- Simcoe, Amy L
- Olsen, David B
- Schleif, William A
- Carella, Anthony
- Gabryelski, Lori
- Jin, Lixia
- Lin, Jiunn H
- Emini, Emilio
- Chapman, Kevin
- Tata, James R
Producer: 20040128
In:
Bioorganic & medicinal chemistry letters vol. 13
Availability: No items available.
|
|
6.
|
Tetrahydro anthranilic acid as a surrogate for anthranilic acid: application to the discovery of potent niacin receptor agonists. [electronic resource] by
- Raghavan, Subharekha
- Tria, G Scott
- Shen, Hong C
- Ding, Fa-Xiang
- Taggart, Andrew K
- Ren, Ning
- Wilsie, Larrisa C
- Krsmanovic, Mihajlo L
- Holt, Tom G
- Wolff, Michael S
- Waters, M Gerard
- Hammond, Milton L
- Tata, James R
- Colletti, Steven L
Producer: 20080709
In:
Bioorganic & medicinal chemistry letters vol. 18
Availability: No items available.
|
|
7.
|
Pyrazole acids as niacin receptor agonists for the treatment of dyslipidemia. [electronic resource] by
- Schmidt, Darby
- Smenton, Abigail
- Raghavan, Subharekha
- Carballo-Jane, Ester
- Lubell, Silvi
- Ciecko, Tanya
- Holt, Tom G
- Wolff, Michael
- Taggart, Andrew
- Wilsie, Larissa
- Krsmanovic, Mihajlo
- Ren, Ning
- Blom, Daniel
- Cheng, Kang
- McCann, Peggy E
- Gerard Waters, M
- Tata, James
- Colletti, Steven
Producer: 20091013
In:
Bioorganic & medicinal chemistry letters vol. 19
Availability: No items available.
|
|
8.
|
GPR109a agonists. Part 1: 5-Alkyl and 5-aryl-pyrazole-tetrazoles as agonists of the human orphan G-protein coupled receptor GPR109a. [electronic resource] by
- Imbriglio, Jason E
- Chang, Sookhee
- Liang, Rui
- Raghavan, Subharekha
- Schmidt, Darby
- Smenton, Abby
- Tria, Scott
- Schrader, Thomas O
- Jung, Jae-Kyu
- Esser, Craig
- Taggart, Andrew K P
- Cheng, Kang
- Carballo-Jane, Ester
- Gerard Waters, M
- Tata, James R
- Colletti, Steven L
Producer: 20090826
In:
Bioorganic & medicinal chemistry letters vol. 19
Availability: No items available.
|
|
9.
|
Anthranilic acid replacements in a niacin receptor agonist. [electronic resource] by
- Schmidt, Darby
- Smenton, Abigail
- Raghavan, Subharekha
- Shen, Hong
- Ding, Fa-Xiang
- Carballo-Jane, Ester
- Luell, Silvi
- Ciecko, Tanya
- Holt, Tom G
- Wolff, Michael
- Taggart, Andrew
- Wilsie, Larissa
- Krsmanovic, Mihajlo
- Ren, Ning
- Blom, Daniel
- Cheng, Kang
- McCann, Peggy E
- Waters, M Gerard
- Tata, James
- Colletti, Steven
Producer: 20100810
In:
Bioorganic & medicinal chemistry letters vol. 20
Availability: No items available.
|
|
10.
|
GPR109a agonists. Part 2: pyrazole-acids as agonists of the human orphan G-protein coupled receptor GPR109a. [electronic resource] by
- Imbriglio, Jason E
- Chang, Sookhee
- Liang, Rui
- Raghavan, Subharekha
- Schmidt, Darby
- Smenton, Abby
- Tria, Scott
- Schrader, Thomas O
- Jung, Jae-Kyu
- Esser, Craig
- Holt, Tom G
- Wolff, Michael S
- Taggart, Andrew K P
- Cheng, Kang
- Carballo-Jane, Ester
- Waters, M Gerard
- Tata, James R
- Colletti, Steven L
Producer: 20101123
In:
Bioorganic & medicinal chemistry letters vol. 20
Availability: No items available.
|
|
11.
|
Discovery of a biaryl cyclohexene carboxylic acid (MK-6892): a potent and selective high affinity niacin receptor full agonist with reduced flushing profiles in animals as a preclinical candidate. [electronic resource] by
- Shen, Hong C
- Ding, Fa-Xiang
- Raghavan, Subharekha
- Deng, Qiaolin
- Luell, Silvi
- Forrest, Michael J
- Carballo-Jane, Ester
- Wilsie, Larissa C
- Krsmanovic, Mihajlo L
- Taggart, Andrew K
- Wu, Kenneth K
- Wu, Tsuei-Ju
- Cheng, Kang
- Ren, Ning
- Cai, Tian-Quan
- Chen, Qing
- Wang, Junying
- Wolff, Michael S
- Tong, Xinchun
- Holt, Tom G
- Waters, M Gerard
- Hammond, Milton L
- Tata, James R
- Colletti, Steven L
Producer: 20100504
In:
Journal of medicinal chemistry vol. 53
Availability: No items available.
|