Results
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1.
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A novel, selective, and efficacious nanomolar pyridopyrazinone inhibitor of V600EBRAF. [electronic resource] by
- Whittaker, Steven
- Ménard, Delphine
- Kirk, Ruth
- Ogilvie, Lesley
- Hedley, Douglas
- Zambon, Alfonso
- Lopes, Filipa
- Preece, Natasha
- Manne, Helen
- Rana, Sareena
- Lambros, Maryou
- Reis-Filho, Jorge S
- Marais, Richard
- Springer, Caroline J
Producer: 20101123
In:
Cancer research vol. 70
Availability: No items available.
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2.
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BRAF inhibitors based on an imidazo[4,5]pyridin-2-one scaffold and a meta substituted middle ring. [electronic resource] by
- Nourry, Arnaud
- Zambon, Alfonso
- Davies, Lawrence
- Niculescu-Duvaz, Ion
- Dijkstra, Harmen P
- Ménard, Delphine
- Gaulon, Catherine
- Niculescu-Duvaz, Dan
- Suijkerbuijk, Bart M J M
- Friedlos, Frank
- Manne, Helen A
- Kirk, Ruth
- Whittaker, Steven
- Marais, Richard
- Springer, Caroline J
Producer: 20100401
In:
Journal of medicinal chemistry vol. 53
Availability: No items available.
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3.
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Novel hinge binder improves activity and pharmacokinetic properties of BRAF inhibitors. [electronic resource] by
- Zambon, Alfonso
- Ménard, Delphine
- Suijkerbuijk, Bart M J M
- Niculescu-Duvaz, Ion
- Whittaker, Steven
- Niculescu-Duvaz, Dan
- Nourry, Arnaud
- Davies, Lawrence
- Manne, Helen A
- Lopes, Filipa
- Preece, Natasha
- Hedley, Douglas
- Ogilvie, Lesley M
- Kirk, Ruth
- Marais, Richard
- Springer, Caroline J
Producer: 20100908
In:
Journal of medicinal chemistry vol. 53
Availability: No items available.
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4.
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Novel potent BRAF inhibitors: toward 1 nM compounds through optimization of the central phenyl ring. [electronic resource] by
- Ménard, Delphine
- Niculescu-Duvaz, Ion
- Dijkstra, Harmen P
- Niculescu-Duvaz, Dan
- Suijkerbuijk, Bart M J M
- Zambon, Alfonso
- Nourry, Arnaud
- Roman, Esteban
- Davies, Lawrence
- Manne, Helen A
- Friedlos, Frank
- Kirk, Ruth
- Whittaker, Steven
- Gill, Adrian
- Taylor, Richard D
- Marais, Richard
- Springer, Caroline J
Producer: 20090812
In:
Journal of medicinal chemistry vol. 52
Availability: No items available.
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5.
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Novel tricyclic pyrazole BRAF inhibitors with imidazole or furan central scaffolds. [electronic resource] by
- Niculescu-Duvaz, Dan
- Niculescu-Duvaz, Ion
- Suijkerbuijk, Bart M J M
- Ménard, Delphine
- Zambon, Alfonso
- Nourry, Arnaud
- Davies, Lawrence
- Manne, Helen A
- Friedlos, Frank
- Ogilvie, Lesley
- Hedley, Douglas
- Takle, Andrew K
- Wilson, David M
- Pons, Jean-Francois
- Coulter, Tom
- Kirk, Ruth
- Cantarino, Neus
- Whittaker, Steven
- Marais, Richard
- Springer, Caroline J
Producer: 20101230
In:
Bioorganic & medicinal chemistry vol. 18
Availability: No items available.
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6.
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Pyridoimidazolones as novel potent inhibitors of v-Raf murine sarcoma viral oncogene homologue B1 (BRAF). [electronic resource] by
- Niculescu-Duvaz, Dan
- Gaulon, Catherine
- Dijkstra, Harmen P
- Niculescu-Duvaz, Ion
- Zambon, Alfonso
- Ménard, Delphine
- Suijkerbuijk, Bart M J M
- Nourry, Arnaud
- Davies, Lawrence
- Manne, Helen
- Friedlos, Frank
- Ogilvie, Lesley
- Hedley, Douglas
- Whittaker, Steven
- Kirk, Ruth
- Gill, Adrian
- Taylor, Richard D
- Raynaud, Florence I
- Moreno-Farre, Javier
- Marais, Richard
- Springer, Caroline J
Producer: 20090506
In:
Journal of medicinal chemistry vol. 52
Availability: No items available.
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7.
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Development of novel, highly potent inhibitors of V-RAF murine sarcoma viral oncogene homologue B1 (BRAF): increasing cellular potency through optimization of a distal heteroaromatic group. [electronic resource] by
- Suijkerbuijk, Bart M J M
- Niculescu-Duvaz, Ion
- Gaulon, Catherine
- Dijkstra, Harmen P
- Niculescu-Duvaz, Dan
- Ménard, Delphine
- Zambon, Alfonso
- Nourry, Arnaud
- Davies, Lawrence
- Manne, Helen A
- Friedlos, Frank
- Ogilvie, Lesley M
- Hedley, Douglas
- Lopes, Filipa
- Preece, Natasha P U
- Moreno-Farre, Javier
- Raynaud, Florence I
- Kirk, Ruth
- Whittaker, Steven
- Marais, Richard
- Springer, Caroline J
Producer: 20100510
In:
Journal of medicinal chemistry vol. 53
Availability: No items available.
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