Receptor localization, native tissue binding and ex vivo occupancy for centrally penetrant P2X7 antagonists in the rat. [electronic resource]
Producer: 20110629Description: 405-14 p. digitalISSN:- 1476-5381
- Animals
- Autoradiography
- Binding, Competitive
- Brain -- metabolism
- Cerebral Cortex -- metabolism
- Drug Discovery
- Guanidines -- blood
- Male
- Molecular Targeted Therapy
- Protein Binding
- Purinergic P2X Receptor Antagonists -- metabolism
- Quinolines -- blood
- Radioligand Assay
- Rats
- Rats, Sprague-Dawley
- Receptors, Purinergic P2X7 -- metabolism
- Spinal Cord -- metabolism
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Publication Type: Journal Article
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