Receptor localization, native tissue binding and ex vivo occupancy for centrally penetrant P2X7 antagonists in the rat.

Able, S L

Receptor localization, native tissue binding and ex vivo occupancy for centrally penetrant P2X7 antagonists in the rat. [electronic resource] - British journal of pharmacology Jan 2011 - 405-14 p. digital

Publication Type: Journal Article

1476-5381

10.1111/j.1476-5381.2010.01025.x doi


Animals
Autoradiography
Binding, Competitive
Brain--metabolism
Cerebral Cortex--metabolism
Drug Discovery
Guanidines--blood
Male
Molecular Targeted Therapy
Protein Binding
Purinergic P2X Receptor Antagonists--metabolism
Quinolines--blood
Radioligand Assay
Rats
Rats, Sprague-Dawley
Receptors, Purinergic P2X7--metabolism
Spinal Cord--metabolism