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Entry into a new class of potent proteasome inhibitors having high antiproliferative activity by structure-based design. [electronic resource] by
- Furet, Pascal
- Imbach, Patricia
- Noorani, Maria
- Koeppler, Juergen
- Laumen, Kurt
- Lang, Marc
- Guagnano, Vito
- Fuerst, Peter
- Roesel, Johannes
- Zimmermann, Johann
- García-Echeverría, Carlos
Producer: 20041101
In:
Journal of medicinal chemistry vol. 47
Availability: No items available.
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2-Amino-aryl-7-aryl-benzoxazoles as potent, selective and orally available JAK2 inhibitors. [electronic resource] by
- Gerspacher, Marc
- Furet, Pascal
- Pissot-Soldermann, Carole
- Gaul, Christoph
- Holzer, Philipp
- Vangrevelinghe, Eric
- Lang, Marc
- Erdmann, Dirk
- Radimerski, Thomas
- Regnier, Catherine H
- Chene, Patrick
- De Pover, Alain
- Hofmann, Francesco
- Baffert, Fabienne
- Buhl, Thomas
- Aichholz, Reiner
- Blasco, Francesca
- Endres, Ralf
- Trappe, Jörg
- Drueckes, Peter
Producer: 20100527
In:
Bioorganic & medicinal chemistry letters vol. 20
Availability: No items available.
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Debio 0617B Inhibits Growth of STAT3-Driven Solid Tumors through Combined Inhibition of JAK, SRC, and Class III/V Receptor Tyrosine Kinases. [electronic resource] by
- Murone, Maximilien
- Vaslin Chessex, Anne
- Attinger, Antoine
- Ramachandra, Raghuveer
- Shetty, Shankar J
- Daginakatte, Girish
- Sengupta, Saumitra
- Marappan, Sivapriya
- Dhodheri, Samiulla
- Rigotti, Stefania
- Bachhav, Yogeshwar
- Brienza, Silvano
- Traxler, Peter
- Lang, Marc
- Aguet, Michel
- Zoete, Vincent
- Michielin, Olivier
- Nicholas, Courtney
- Johnson, Faye M
- Ramachandra, Murali
- McAllister, Andres
Producer: 20170615
In:
Molecular cancer therapeutics vol. 15
Availability: No items available.
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Potent and selective inhibition of polycythemia by the quinoxaline JAK2 inhibitor NVP-BSK805. [electronic resource] by
- Baffert, Fabienne
- Régnier, Catherine H
- De Pover, Alain
- Pissot-Soldermann, Carole
- Tavares, Gisele A
- Blasco, Francesca
- Brueggen, Josef
- Chène, Patrick
- Drueckes, Peter
- Erdmann, Dirk
- Furet, Pascal
- Gerspacher, Marc
- Lang, Marc
- Ledieu, David
- Nolan, Lynda
- Ruetz, Stephan
- Trappe, Joerg
- Vangrevelinghe, Eric
- Wartmann, Markus
- Wyder, Lorenza
- Hofmann, Francesco
- Radimerski, Thomas
Producer: 20101104
In:
Molecular cancer therapeutics vol. 9
Availability: No items available.
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