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Synthesis of water-soluble (aminoalkyl)camptothecin analogues: inhibition of topoisomerase I and antitumor activity. [electronic resource] by
- Kingsbury, W D
- Boehm, J C
- Jakas, D R
- Holden, K G
- Hecht, S M
- Gallagher, G
- Caranfa, M J
- McCabe, F L
- Faucette, L F
- Johnson, R K
Producer: 19910312
In:
Journal of medicinal chemistry vol. 34
Availability: No items available.
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Modification of the hydroxy lactone ring of camptothecin: inhibition of mammalian topoisomerase I and biological activity. [electronic resource] by
- Hertzberg, R P
- Caranfa, M J
- Holden, K G
- Jakas, D R
- Gallagher, G
- Mattern, M R
- Mong, S M
- Bartus, J O
- Johnson, R K
- Kingsbury, W D
Producer: 19890406
In:
Journal of medicinal chemistry vol. 32
Availability: No items available.
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7.
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(E)-3-[[[[6-(2-carboxyethenyl)-5-[[8-(4- methoxyphenyl)octyl]oxy]-2-pyridinyl]-methyl]thio]methyl]benzoic acid and related compounds: high affinity leukotriene B4 receptor antagonists. [electronic resource] by
- Daines, R A
- Chambers, P A
- Eggleston, D S
- Foley, J J
- Griswold, D E
- Haltiwanger, R C
- Jakas, D R
- Kingsbury, W D
- Martin, L D
- Pendrak, I
Producer: 19941103
In:
Journal of medicinal chemistry vol. 37
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8.
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(E)-3-[[[[6-(2-carboxyethenyl)-5-[[8-(4- methoxyphenyl)octyl]oxy]-2-pyridinyl]-methyl]thio]methyl]benzoic acid: a novel high-affinity leukotriene B4 receptor antagonist. [electronic resource] by
- Daines, R A
- Chambers, P A
- Pendrak, I
- Jakas, D R
- Sarau, H M
- Foley, J J
- Schmidt, D B
- Griswold, D E
- Martin, L D
- Tzimas, M N
Producer: 19931029
In:
Journal of medicinal chemistry vol. 36
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9.
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Orally active 7-phenylglycyl cephalosporins. Structure-activity studies related to cefatrizine (SK&F 60771). [electronic resource] by
- Dunn, G L
- Hoover, J R
- Berges, D A
- Taggart, J J
- Davis, L D
- Dietz, E M
- Jakas, D R
- Yim, N
- Actor, P
- Uri, J V
- Weisbach, J A
Producer: 19760901
In:
The Journal of antibiotics vol. 29
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10.
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Preclinical pharmacokinetics and interspecies scaling of a novel vitronectin receptor antagonist. [electronic resource] by
- Ward, K W
- Azzarano, L M
- Bondinell, W E
- Cousins, R D
- Huffman, W F
- Jakas, D R
- Keenan, R M
- Ku, T W
- Lundberg, D
- Miller, W H
- Mumaw, J A
- Newlander, K A
- Pirhalla, J L
- Roethke, T J
- Salyers, K L
- Souder, P R
- Stelman, G J
- Smith, B R
Producer: 19991124
In:
Drug metabolism and disposition: the biological fate of chemicals vol. 27
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11.
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In vitro and in vivo pharmacological characterization of SB 201993, an eicosanoid-like LTB4 receptor antagonist with anti-inflammatory activity. [electronic resource] by
- Sarau, H M
- Foley, J J
- Schmidt, D B
- Martin, L D
- Webb, E F
- Tzimas, M N
- Breton, J J
- Chabot-Fletcher, M
- Underwood, D C
- Hay, D W
- Kingsbury, W D
- Chambers, P A
- Pendrak, I
- Jakas, D R
- Sathe, G M
- Van Horn, S
- Daines, R A
- Griswold, D E
Producer: 19991007
In:
Prostaglandins, leukotrienes, and essential fatty acids vol. 61
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12.
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Discovery of an imidazopyridine-containing 1,4-benzodiazepine nonpeptide vitronectin receptor (alpha v beta 3) antagonist with efficacy in a restenosis model. [electronic resource] by
- Keenan, R M
- Lago, M A
- Miller, W H
- Ali, F E
- Cousins, R D
- Hall, L B
- Hwang, S M
- Jakas, D R
- Kwon, C
- Louden, C
- Nguyen, T T
- Ohlstein, E H
- Rieman, D J
- Ross, S T
- Samanen, J M
- Smith, B R
- Stadel, J
- Takata, D T
- Vickery, L
- Yuan, C C
- Yue, T L
Producer: 19990126
In:
Bioorganic & medicinal chemistry letters vol. 8
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13.
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Benzimidazole derivatives as arginine mimetics in 1,4-benzodiazepine nonpeptide vitronectin receptor (alpha v beta 3) antagonists. [electronic resource] by
- Keenan, R M
- Miller, W H
- Lago, M A
- Ali, F E
- Bondinell, W E
- Callahan, J F
- Calvo, R R
- Cousins, R D
- Hwang, S M
- Jakas, D R
- Ku, T W
- Kwon, C
- Nguyen, T T
- Reader, V A
- Rieman, D J
- Ross, S T
- Takata, D T
- Uzinskas, I N
- Yuan, C C
- Smith, B R
Producer: 19990126
In:
Bioorganic & medicinal chemistry letters vol. 8
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14.
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Conformational preferences in a benzodiazepine series of potent nonpeptide fibrinogen receptor antagonists. [electronic resource] by
- Keenan, R M
- Callahan, J F
- Samanen, J M
- Bondinell, W E
- Calvo, R R
- Chen, L
- DeBrosse, C
- Eggleston, D S
- Haltiwanger, R C
- Hwang, S M
- Jakas, D R
- Ku, T W
- Miller, W H
- Newlander, K A
- Nichols, A
- Parker, M F
- Southhall, L S
- Uzinskas, I
- Vasko-Moser, J A
- Venslavsky, J W
- Wong, A S
- Huffman, W F
Producer: 19990316
In:
Journal of medicinal chemistry vol. 42
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15.
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Orally bioavailable nonpeptide vitronectin receptor antagonists with efficacy in an osteoporosis model. [electronic resource] by
- Miller, W H
- Bondinell, W E
- Cousins, R D
- Erhard, K F
- Jakas, D R
- Keenan, R M
- Ku, T W
- Newlander, K A
- Ross, S T
- Haltiwanger, R C
- Bradbeer, J
- Drake, F H
- Gowen, M
- Hoffman, S J
- Hwang, S M
- James, I E
- Lark, M W
- Lechowska, B
- Rieman, D J
- Stroup, G B
- Vasko-Moser, J A
- Zembryki, D L
- Azzarano, L M
- Adams, P C
- Huffman, W F
Producer: 19991014
In:
Bioorganic & medicinal chemistry letters vol. 9
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16.
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Potent, selective, orally active 3-oxo-1,4-benzodiazepine GPIIb/IIIa integrin antagonists. [electronic resource] by
- Samanen, J M
- Ali, F E
- Barton, L S
- Bondinell, W E
- Burgess, J L
- Callahan, J F
- Calvo, R R
- Chen, W
- Chen, L
- Erhard, K
- Feuerstein, G
- Heys, R
- Hwang, S M
- Jakas, D R
- Keenan, R M
- Ku, T W
- Kwon, C
- Lee, C P
- Miller, W H
- Newlander, K A
- Nichols, A
- Parker, M
- Peishoff, C E
- Rhodes, G
- Ross, S
- Shu, A
- Simpson, R
- Takata, D
- Yellin, T O
- Uzsinskas, I
- Venslavsky, J W
- Yuan, C K
- Huffman, W F
Producer: 19970123
In:
Journal of medicinal chemistry vol. 39
Availability: No items available.
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