Results
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Discovery of furo[2,3-d][1,3]thiazinamines as beta amyloid cleaving enzyme-1 (BACE1) inhibitors. [electronic resource] by
- Wu, Yong-Jin
- Guernon, Jason
- Rajamani, Ramkumar
- Toyn, Jeremy H
- Ahlijanian, Michael K
- Albright, Charles F
- Muckelbauer, Jodi
- Chang, ChiehYing
- Camac, Dan
- Macor, John E
- Thompson, Lorin A
Producer: 20170627
In:
Bioorganic & medicinal chemistry letters vol. 26
Availability: No items available.
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3.
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3-Thio-quinolinone maxi-K openers for the treatment of erectile dysfunction. [electronic resource] by
- Boy, Kenneth M
- Guernon, Jason M
- Sit, Sing-Yuen
- Xie, Kai
- Hewawasam, Piyasena
- Boissard, Christopher G
- Dworetzky, Steven I
- Natale, Joanne
- Gribkoff, Valentin K
- Lodge, Nicholas
- Starrett, John E
Producer: 20050404
In:
Bioorganic & medicinal chemistry letters vol. 14
Availability: No items available.
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4.
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Discovery of new indole-based acylsulfonamide Na [electronic resource] by
- Wu, Yong-Jin
- Venables, Brian
- Guernon, Jason
- Chen, Jie
- Sit, Sing-Yuen
- Rajamani, Ramkumar
- Knox, Ronald J
- Matchett, Michele
- Pieschl, Rick L
- Herrington, James
- Bristow, Linda J
- Meanwell, Nicholas A
- Thompson, Lorin A
- Dzierba, Carolyn
Producer: 20200305
In:
Bioorganic & medicinal chemistry letters vol. 29
Availability: No items available.
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5.
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Discovery of S3-Truncated, C-6 Heteroaryl Substituted Aminothiazine β-Site APP Cleaving Enzyme-1 (BACE1) Inhibitors. [electronic resource] by
- Wu, Yong-Jin
- Guernon, Jason
- Shi, Jianliang
- Marcin, Lawrence
- Higgins, Mendi
- Rajamani, Ramkumar
- Muckelbauer, Jodi
- Lewis, Hal
- Chang, ChiehYing
- Camac, Dan
- Toyn, Jeremy H
- Ahlijanian, Michael K
- Albright, Charles F
- Macor, John E
- Thompson, Lorin A
Producer: 20170612
In:
Journal of medicinal chemistry vol. 59
Availability: No items available.
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6.
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Discovery of morpholine-based aryl sulfonamides as Na [electronic resource] by
- Wu, Yong-Jin
- Guernon, Jason
- McClure, Andrea
- Venables, Brian
- Rajamani, Ramkumar
- Robbins, Kevin J
- Knox, Ronald J
- Matchett, Michele
- Pieschl, Rick L
- Herrington, James
- Bristow, Linda J
- Meanwell, Nicholas A
- Olson, Richard
- Thompson, Lorin A
- Dzierba, Carolyn
Producer: 20181002
In:
Bioorganic & medicinal chemistry letters vol. 28
Availability: No items available.
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7.
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Targeting the BACE1 Active Site Flap Leads to a Potent Inhibitor That Elicits Robust Brain Aβ Reduction in Rodents. [electronic resource] by
- Wu, Yong-Jin
- Guernon, Jason
- Yang, Fukang
- Snyder, Lawrence
- Shi, Jianliang
- Mcclure, Andrea
- Rajamani, Ramkumar
- Park, Hyunsoo
- Ng, Alicia
- Lewis, Hal
- Chang, ChiehYing
- Camac, Dan
- Toyn, Jeremy H
- Ahlijanian, Michael K
- Albright, Charles F
- Macor, John E
- Thompson, Lorin A
Producer: 20160317
In:
ACS medicinal chemistry letters vol. 7
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8.
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Monosubstituted γ-lactam and conformationally constrained 1,3-diaminopropan-2-ol transition-state isostere inhibitors of β-secretase (BACE). [electronic resource] by
- Boy, Kenneth M
- Guernon, Jason M
- Shi, Jianliang
- Toyn, Jeremy H
- Meredith, Jere E
- Barten, Donna M
- Burton, Catherine R
- Albright, Charles F
- Marcinkeviciene, Jovita
- Good, Andrew C
- Tebben, Andrew J
- Muckelbauer, Jodi K
- Camac, Daniel M
- Lentz, Kimberley A
- Bronson, Joanne J
- Olson, Richard E
- Macor, John E
- Thompson, Lorin A
Producer: 20120213
In:
Bioorganic & medicinal chemistry letters vol. 21
Availability: No items available.
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9.
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Macrocyclic prolinyl acyl guanidines as inhibitors of β-secretase (BACE). [electronic resource] by
- Boy, Kenneth M
- Guernon, Jason M
- Wu, Yong-Jin
- Zhang, Yunhui
- Shi, Joe
- Zhai, Weixu
- Zhu, Shirong
- Gerritz, Samuel W
- Toyn, Jeremy H
- Meredith, Jere E
- Barten, Donna M
- Burton, Catherine R
- Albright, Charles F
- Good, Andrew C
- Grace, James E
- Lentz, Kimberley A
- Olson, Richard E
- Macor, John E
- Thompson, Lorin A
Producer: 20160811
In:
Bioorganic & medicinal chemistry letters vol. 25
Availability: No items available.
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10.
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Development of New Benzenesulfonamides As Potent and Selective Na [electronic resource] by
- Wu, Yong-Jin
- Guernon, Jason
- Shi, Jianliang
- Ditta, Jonathan
- Robbins, Kevin J
- Rajamani, Ramkumar
- Easton, Amy
- Newton, Amy
- Bourin, Clotilde
- Mosure, Kathleen
- Soars, Matthew G
- Knox, Ronald J
- Matchett, Michele
- Pieschl, Rick L
- Post-Munson, Debra J
- Wang, Shuya
- Herrington, James
- Graef, John
- Newberry, Kimberly
- Bristow, Linda J
- Meanwell, Nicholas A
- Olson, Richard
- Thompson, Lorin A
- Dzierba, Carolyn
Producer: 20170619
In:
Journal of medicinal chemistry vol. 60
Availability: No items available.
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11.
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Discovery of non-zwitterionic aryl sulfonamides as Na [electronic resource] by
- Wu, Yong-Jin
- Guernon, Jason
- McClure, Andrea
- Luo, Guanglin
- Rajamani, Ramkumar
- Ng, Alicia
- Easton, Amy
- Newton, Amy
- Bourin, Clotilde
- Parker, Dawn
- Mosure, Kathleen
- Barnaby, Omar
- Soars, Matthew G
- Knox, Ronald J
- Matchett, Michele
- Pieschl, Rick
- Herrington, James
- Chen, Ping
- Sivarao, D V
- Bristow, Linda J
- Meanwell, Nicholas A
- Bronson, Joanne
- Olson, Richard
- Thompson, Lorin A
- Dzierba, Carolyn
Producer: 20171108
In:
Bioorganic & medicinal chemistry vol. 25
Availability: No items available.
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12.
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The discovery of VU0652957 (VU2957, Valiglurax): SAR and DMPK challenges en route to an mGlu [electronic resource] by
- Panarese, Joseph D
- Engers, Darren W
- Wu, Yong-Jin
- Guernon, Jason M
- Chun, Aspen
- Gregro, Alison R
- Bender, Aaron M
- Capstick, Rory A
- Wieting, Joshua M
- Bronson, Joanne J
- Macor, John E
- Westphal, Ryan
- Soars, Matthew
- Engers, Julie E
- Felts, Andrew S
- Rodriguez, Alice L
- Emmitte, Kyle A
- Jones, Carrie K
- Blobaum, Anna L
- Conn, P Jeffrey
- Niswender, Colleen M
- Hopkins, Corey R
- Lindsley, Craig W
Producer: 20191104
In:
Bioorganic & medicinal chemistry letters vol. 29
Availability: No items available.
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13.
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Synthesis and in vivo evaluation of cyclic diaminopropane BACE-1 inhibitors. [electronic resource] by
- Thompson, Lorin A
- Shi, Jianliang
- Decicco, Carl P
- Tebben, Andrew J
- Olson, Richard E
- Boy, Kenneth M
- Guernon, Jason M
- Good, Andrew C
- Liauw, Ann
- Zheng, Changsheng
- Copeland, Robert A
- Combs, Andrew P
- Trainor, George L
- Camac, Daniel M
- Muckelbauer, Jodi K
- Lentz, Kimberley A
- Grace, James E
- Burton, Catherine R
- Toyn, Jeremy H
- Barten, Donna M
- Marcinkeviciene, Jovita
- Meredith, Jere E
- Albright, Charles F
- Macor, John E
Producer: 20120213
In:
Bioorganic & medicinal chemistry letters vol. 21
Availability: No items available.
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14.
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Identification and Preclinical Evaluation of the Bicyclic Pyrimidine γ-Secretase Modulator BMS-932481. [electronic resource] by
- Boy, Kenneth M
- Guernon, Jason M
- Zuev, Dmitry S
- Xu, Li
- Zhang, Yunhui
- Shi, Jianliang
- Marcin, Lawrence R
- Higgins, Mendi A
- Wu, Yong-Jin
- Krishnananthan, Subramaniam
- Li, Jianqing
- Trehan, Ashok
- Smith, Daniel
- Toyn, Jeremy H
- Meredith, Jere E
- Burton, Catherine R
- Kimura, S Roy
- Zvyaga, Tatyana
- Zhuo, Xiaoliang
- Lentz, Kimberley A
- Grace, James E
- Denton, Rex
- Morrison, John S
- Mathur, Arvind
- Albright, Charles F
- Ahlijanian, Michael K
- Olson, Richard E
- Thompson, Lorin A
- Macor, John E
Publication details: ACS medicinal chemistry letters Mar 2019
In:
ACS medicinal chemistry letters vol. 10
Availability: No items available.
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