Results
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1.
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Stimulation of Glucose-Dependent Insulin Secretion by a Potent, Selective sst3 Antagonist. [electronic resource] by
- Pasternak, Alexander
- Feng, Zhe
- de Jesus, Reynalda
- Ye, Zhixiong
- He, Shuwen
- Dobbelaar, Peter
- Bradley, Scott A
- Chicchi, Gary G
- Tsao, Kwei-Lan
- Trusca, Dorina
- Eiermann, George J
- Li, Cai
- Feng, Yue
- Wu, Margaret
- Shao, Qing
- Zhang, Bei B
- Nargund, Ravi
- Mills, Sander G
- Howard, Andrew D
- Yang, Lihu
- Zhou, Yun-Ping
Producer: 20140605
In:
ACS medicinal chemistry letters vol. 3
Availability: No items available.
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2.
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Spiroindane based amides as potent and selective MC4R agonists for the treatment of obesity. [electronic resource] by
- He, Shuwen
- Ye, Zhixiong
- Dobbelaar, Peter H
- Sebhat, Iyassu K
- Guo, Liangqin
- Liu, Jian
- Jian, Tianying
- Lai, Yingjie
- Franklin, Christopher L
- Bakshi, Raman K
- Dellureficio, James P
- Hong, Qingmei
- Weinberg, David H
- Macneil, Tanya
- Tang, Rui
- Strack, Alison M
- Tamvakopoulos, Constantin
- Peng, Qianping
- Miller, Randy R
- Stearns, Ralph A
- Chen, Howard Y
- Chen, Airu S
- Fong, Tung M
- Wyvratt, Matthew J
- Nargund, Ravi P
Producer: 20101123
In:
Bioorganic & medicinal chemistry letters vol. 20
Availability: No items available.
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3.
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Discovery of potent, selective, and orally bioavailable 3H-spiro[isobenzofuran-1,4'-piperidine] based melanocortin subtype-4 receptor agonists. [electronic resource] by
- Guo, Liangqin
- Ye, Zhixiong
- Liu, Jian
- He, Shuwen
- Bakshi, Raman K
- Sebhat, Iyassu K
- Dobbelaar, Peter H
- Hong, Qingmei
- Jian, Tianying
- Dellureficio, James P
- Tsou, Nancy N
- Ball, Richard G
- Weinberg, David H
- MacNeil, Tanya
- Tang, Rui
- Tamvakopoulos, Constantin
- Peng, Qianping
- Chen, Howard Y
- Chen, Airu S
- Martin, William J
- MacIntyre, D Euan
- Strack, Alison M
- Fong, Tung M
- Wyvratt, Matthew J
- Nargund, Ravi P
Producer: 20101110
In:
Bioorganic & medicinal chemistry letters vol. 20
Availability: No items available.
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4.
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Discovery of highly potent and efficacious MC4R agonists with spiroindane N-Me-1,2,4-triazole privileged structures for the treatment of obesity. [electronic resource] by
- He, Shuwen
- Ye, Zhixiong
- Dobbelaar, Peter H
- Bakshi, Raman K
- Hong, Qingmei
- Dellureficio, James P
- Sebhat, Iyassu K
- Guo, Liangqin
- Liu, Jian
- Jian, Tianying
- Lai, Yingjie
- Franklin, Christopher L
- Reibarkh, Mikhail
- Holmes, Mark A
- Weinberg, David H
- MacNeil, Tanya
- Tang, Rui
- Tamvakopoulos, Constantin
- Peng, Qianping
- Miller, Randy R
- Stearns, Ralph A
- Chen, Howard Y
- Chen, Airu S
- Strack, Alison M
- Fong, Tung M
- Wyvratt, Matthew J
- Nargund, Ravi P
Producer: 20110329
In:
Bioorganic & medicinal chemistry letters vol. 20
Availability: No items available.
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5.
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Synthesis and SAR of derivatives based on 2-biarylethylimidazole as bombesin receptor subtype-3 (BRS-3) agonists for the treatment of obesity. [electronic resource] by
- Liu, Jian
- He, Shuwen
- Jian, Tianying
- Dobbelaar, Peter H
- Sebhat, Iyassu K
- Lin, Linus S
- Goodman, Allan
- Guo, Cheng
- Guzzo, Peter R
- Hadden, Mark
- Henderson, Alan J
- Pattamana, Kevin
- Ruenz, Megan
- Sargent, Bruce J
- Swenson, Brian
- Yet, Larry
- Tamvakopoulos, Constantin
- Peng, Qianping
- Pan, Jie
- Kan, Yanqing
- Palyha, Oksana
- Kelly, Theresa M
- Guan, Xiao-Ming
- Howard, Andrew D
- Marsh, Donald J
- Metzger, Joseph M
- Reitman, Marc L
- Wyvratt, Matthew J
- Nargund, Ravi P
Producer: 20100705
In:
Bioorganic & medicinal chemistry letters vol. 20
Availability: No items available.
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6.
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Regulation of energy homeostasis by bombesin receptor subtype-3: selective receptor agonists for the treatment of obesity. [electronic resource] by
- Guan, Xiao-Ming
- Chen, Howard
- Dobbelaar, Peter H
- Dong, Yan
- Fong, Tung M
- Gagen, Karen
- Gorski, Judith
- He, Shuwen
- Howard, Andrew D
- Jian, Tianying
- Jiang, Michael
- Kan, Yanqing
- Kelly, Theresa M
- Kosinski, Jennifer
- Lin, Linus S
- Liu, Jian
- Marsh, Donald J
- Metzger, Joseph M
- Miller, Randy
- Nargund, Ravi P
- Palyha, Oksana
- Shearman, Lauren
- Shen, Zhu
- Stearns, Ralph
- Strack, Alison M
- Stribling, Sloan
- Tang, Yui Sing
- Wang, Sheng-Ping
- White, Amanda
- Yu, Hong
- Reitman, Marc L
Producer: 20100429
In:
Cell metabolism vol. 11
Availability: No items available.
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7.
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Discovery of a spiroindane based compound as a potent, selective, orally bioavailable melanocortin subtype-4 receptor agonist. [electronic resource] by
- He, Shuwen
- Ye, Zhixiong
- Dobbelaar, Peter H
- Sebhat, Iyassu K
- Guo, Liangqin
- Liu, Jian
- Jian, Tianying
- Lai, Yingjie
- Franklin, Christopher L
- Bakshi, Raman K
- Dellureficio, James P
- Hong, Qingmei
- Tsou, Nancy N
- Ball, Richard G
- Cashen, Doreen E
- Martin, William J
- Weinberg, David H
- Macneil, Tanya
- Tang, Rui
- Tamvakopoulos, Constantin
- Peng, Qianping
- Miller, Randy R
- Stearns, Ralph A
- Chen, Howard Y
- Chen, Airu S
- Strack, Alison M
- Fong, Tung M
- Macintyre, D Euan
- Wyvratt, Matthew J
- Nargund, Ravi P
Producer: 20100705
In:
Bioorganic & medicinal chemistry letters vol. 20
Availability: No items available.
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8.
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Optimization of privileged structures for selective and potent melanocortin subtype-4 receptor ligands. [electronic resource] by
- Hong, Qingmei
- Bakshi, Raman K
- Dellureficio, James
- He, Shuwen
- Ye, Zhixiong
- Dobbelaar, Peter H
- Sebhat, Iyassu K
- Guo, Liangqin
- Liu, Jian
- Jian, Tianying
- Tang, Rui
- Kalyani, Rubana N
- Macneil, Tanya
- Vongs, Aurawan
- Rosenblum, Charles I
- Weinberg, David H
- Peng, Qingping
- Tamvakopoulos, Constantin
- Miller, Randy R
- Stearns, Ralph A
- Cashen, Doreen
- Martin, Willian J
- Chen, Airu S
- Metzger, Joseph M
- Chen, Howard Y
- Strack, Allison M
- Fong, Tung M
- Maclntyre, Euan
- Van der Ploeg, Lex H T
- Wyvratt, Matthew J
- Nargund, Ravi P
Producer: 20101123
In:
Bioorganic & medicinal chemistry letters vol. 20
Availability: No items available.
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9.
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Discovery of substituted biphenyl imidazoles as potent, bioavailable bombesin receptor subtype-3 agonists. [electronic resource] by
- He, Shuwen
- Dobbelaar, Peter H
- Liu, Jian
- Jian, Tianying
- Sebhat, Iyassu K
- Lin, Linus S
- Goodman, Allan
- Guo, Cheng
- Guzzo, Peter R
- Hadden, Mark
- Henderson, Alan J
- Ruenz, Megan
- Sargent, Bruce J
- Yet, Larry
- Kelly, Theresa M
- Palyha, Oksana
- Kan, Yanqing
- Pan, Jie
- Chen, Howard
- Marsh, Donald J
- Shearman, Lauren P
- Strack, Alison M
- Metzger, Joseph M
- Feighner, Scott D
- Tan, Carina
- Howard, Andrew D
- Tamvakopoulos, Constantin
- Peng, Qianping
- Guan, Xiao-Ming
- Reitman, Marc L
- Patchett, Arthur A
- Wyvratt, Matthew J
- Nargund, Ravi P
Producer: 20100713
In:
Bioorganic & medicinal chemistry letters vol. 20
Availability: No items available.
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10.
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Investigation of Cardiovascular Effects of Tetrahydro-β-carboline sstr3 antagonists. [electronic resource] by
- He, Shuwen
- Lai, Zhong
- Ye, Zhixiong
- Dobbelaar, Peter H
- Shah, Shrenik K
- Truong, Quang
- Du, Wu
- Guo, Liangqin
- Liu, Jian
- Jian, Tianying
- Qi, Hongbo
- Bakshi, Raman K
- Hong, Qingmei
- Dellureficio, James
- Reibarkh, Mikhail
- Samuel, Koppara
- Reddy, Vijay B
- Mitelman, Stan
- Tong, Sharon X
- Chicchi, Gary G
- Tsao, Kwei-Lan
- Trusca, Dorina
- Wu, Margaret
- Shao, Qing
- Trujillo, Maria E
- Fernandez, Guillermo
- Nelson, Donald
- Bunting, Patricia
- Kerr, Janet
- Fitzgerald, Patrick
- Morissette, Pierre
- Volksdorf, Sylvia
- Eiermann, George J
- Li, Cai
- Zhang, Bei
- Howard, Andrew D
- Zhou, Yun-Ping
- Nargund, Ravi P
- Hagmann, William K
Producer: 20140722
In:
ACS medicinal chemistry letters vol. 5
Availability: No items available.
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11.
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SAR exploration at the C-3 position of tetrahydro-β-carboline sstr3 antagonists. [electronic resource] by
- He, Shuwen
- Dobbelaar, Peter H
- Guo, Liangqin
- Ye, Zhixiong
- Liu, Jian
- Jian, Tianying
- Truong, Quang
- Shah, Shrenik K
- Du, Wu
- Qi, Hongbo
- Bakshi, Raman K
- Hong, Qingmei
- Dellureficio, James D
- Sherer, Edward
- Pasternak, Alexander
- Feng, Zhe
- Reibarkh, Mikhail
- Lin, Melissa
- Samuel, Koppara
- Reddy, Vijay B
- Mitelman, Stan
- Tong, Sharon X
- Chicchi, Gary G
- Tsao, Kwei-Lan
- Trusca, Dorina
- Wu, Margaret
- Shao, Qing
- Trujillo, Maria E
- Fernandez, Guillermo
- Nelson, Donald
- Bunting, Patricia
- Kerr, Janet
- Fitzgerald, Patrick
- Morissette, Pierre
- Volksdorf, Sylvia
- Eiermann, George J
- Li, Cai
- Zhang, Bei B
- Howard, Andrew D
- Zhou, Yun-Ping
- Nargund, Ravi P
- Hagmann, William K
Producer: 20161107
In:
Bioorganic & medicinal chemistry letters vol. 26
Availability: No items available.
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12.
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Discovery of MK-1421, a Potent, Selective sstr3 Antagonist, as a Development Candidate for Type 2 Diabetes. [electronic resource] by
- Shah, Shrenik K
- He, Shuwen
- Guo, Liangqin
- Truong, Quang
- Qi, Hongbo
- Du, Wu
- Lai, Zhong
- Liu, Jian
- Jian, Tianying
- Hong, Qingmei
- Dobbelaar, Peter
- Ye, Zhixiong
- Sherer, Edward
- Feng, Zhe
- Yu, Yang
- Wong, Frederick
- Samuel, Koppara
- Madiera, Maria
- Karanam, Bindhu V
- Reddy, Vijay B
- Mitelman, Stan
- Tong, Sharon X
- Chicchi, Gary G
- Tsao, Kwei-Lan
- Trusca, Dorina
- Feng, Yue
- Wu, Margaret
- Shao, Qing
- Trujillo, Maria E
- Eiermann, George J
- Li, Cai
- Pachanski, Michele
- Fernandez, Guillermo
- Nelson, Donald
- Bunting, Patricia
- Morissette, Pierre
- Volksdorf, Sylvia
- Kerr, Janet
- Zhang, Bei B
- Howard, Andrew D
- Zhou, Yun-Ping
- Pasternak, Alexander
- Nargund, Ravi P
- Hagmann, William K
Producer: 20150525
In:
ACS medicinal chemistry letters vol. 6
Availability: No items available.
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13.
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The Discovery of MK-4256, a Potent SSTR3 Antagonist as a Potential Treatment of Type 2 Diabetes. [electronic resource] by
- He, Shuwen
- Ye, Zhixiong
- Truong, Quang
- Shah, Shrenik
- Du, Wu
- Guo, Liangqin
- Dobbelaar, Peter H
- Lai, Zhong
- Liu, Jian
- Jian, Tianying
- Qi, Hongbo
- Bakshi, Raman K
- Hong, Qingmei
- Dellureficio, James
- Pasternak, Alexander
- Feng, Zhe
- deJesus, Reynalda
- Yang, Lihu
- Reibarkh, Mikhail
- Bradley, Scott A
- Holmes, Mark A
- Ball, Richard G
- Ruck, Rebecca T
- Huffman, Mark A
- Wong, Frederick
- Samuel, Koppara
- Reddy, Vijay B
- Mitelman, Stan
- Tong, Sharon X
- Chicchi, Gary G
- Tsao, Kwei-Lan
- Trusca, Dorina
- Wu, Margaret
- Shao, Qing
- Trujillo, Maria E
- Eiermann, George J
- Li, Cai
- Zhang, Bei B
- Howard, Andrew D
- Zhou, Yun-Ping
- Nargund, Ravi P
- Hagmann, William K
Producer: 20140605
In:
ACS medicinal chemistry letters vol. 3
Availability: No items available.
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