Results
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1.
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2-Benzenesulfonyl-8a-benzyl-hexahydro-2H-isoquinolin-6-ones as selective glucocorticoid receptor antagonists. [electronic resource] by
- Clark, Robin D
- Ray, Nicholas C
- Blaney, Paul
- Crackett, Peter H
- Hurley, Christopher
- Williams, Karen
- Dyke, Hazel J
- Clark, David E
- Lockey, Peter M
- Devos, Rene
- Wong, Melanie
- White, Anne
- Belanoff, Joseph K
Producer: 20071212
In:
Bioorganic & medicinal chemistry letters vol. 17
Availability: No items available.
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2.
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Discovery and optimization of novel, non-steroidal glucocorticoid receptor modulators. [electronic resource] by
- Ray, Nicholas C
- Clark, Robin D
- Clark, David E
- Williams, Karen
- Hickin, H G
- Crackett, Peter H
- Dyke, Hazel J
- Lockey, Peter M
- Wong, Melanie
- Devos, René
- White, Anne
- Belanoff, Joseph K
Producer: 20071120
In:
Bioorganic & medicinal chemistry letters vol. 17
Availability: No items available.
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3.
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Identification and optimisation of a series of substituted 5-(1H-pyrazol-3-yl)-thiophene-2-hydroxamic acids as potent histone deacetylase (HDAC) inhibitors. [electronic resource] by
- Price, Steve
- Bordogna, Walter
- Bull, Richard J
- Clark, David E
- Crackett, Peter H
- Dyke, Hazel J
- Gill, Matthew
- Harris, Neil V
- Gorski, Julia
- Lloyd, Julia
- Lockey, Peter M
- Mullett, Julia
- Roach, Alan G
- Roussel, Fabien
- White, Anne B
Producer: 20070409
In:
Bioorganic & medicinal chemistry letters vol. 17
Availability: No items available.
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4.
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1H-Pyrazolo[3,4-g]hexahydro-isoquinolines as selective glucocorticoid receptor antagonists with high functional activity. [electronic resource] by
- Clark, Robin D
- Ray, Nicholas C
- Williams, Karen
- Blaney, Paul
- Ward, Stuart
- Crackett, Peter H
- Hurley, Christopher
- Dyke, Hazel J
- Clark, David E
- Lockey, Peter
- Devos, Rene
- Wong, Melanie
- Porres, Soraya S
- Bright, Colin P
- Jenkins, Robert E
- Belanoff, Joseph
Producer: 20080512
In:
Bioorganic & medicinal chemistry letters vol. 18
Availability: No items available.
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5.
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Design, synthesis and characterization of a novel class of coumarin-based inhibitors of inducible nitric oxide synthase. [electronic resource] by
- Jackson, Sharon A
- Sahni, Sukhveen
- Lee, Lan
- Luo, Yongyi
- Nieduzak, Thaddeus R
- Liang, Guyan
- Chiang, Yulin
- Collar, Nicola
- Fink, David
- He, Wei
- Laoui, Abdelazize
- Merrill, Jean
- Boffey, Ray
- Crackett, Peter
- Rees, Bryan
- Wong, Melanie
- Guilloteau, Jean-Pierre
- Mathieu, Magali
- Rebello, Sam S
Producer: 20050919
In:
Bioorganic & medicinal chemistry vol. 13
Availability: No items available.
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6.
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Mitigation of Acetylcholine Esterase Activity in the 1,7-Diazacarbazole Series of Inhibitors of Checkpoint Kinase 1. [electronic resource] by
- Gazzard, Lewis
- Williams, Karen
- Chen, Huifen
- Axford, Lorraine
- Blackwood, Elizabeth
- Burton, Brenda
- Chapman, Kerry
- Crackett, Peter
- Drobnick, Joy
- Ellwood, Charles
- Epler, Jennifer
- Flagella, Michael
- Gancia, Emanuela
- Gill, Matthew
- Goodacre, Simon
- Halladay, Jason
- Hewitt, Joanne
- Hunt, Hazel
- Kintz, Samuel
- Lyssikatos, Joseph
- Macleod, Calum
- Major, Sarah
- Médard, Guillaume
- Narukulla, Raman
- Ramiscal, Judi
- Schmidt, Stephen
- Seward, Eileen
- Wiesmann, Christian
- Wu, Ping
- Yee, Sharon
- Yen, Ivana
- Malek, Shiva
Producer: 20150914
In:
Journal of medicinal chemistry vol. 58
Availability: No items available.
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7.
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Novel triazolo-pyrrolopyridines as inhibitors of Janus kinase 1. [electronic resource] by
- Hurley, Christopher A
- Blair, Wade S
- Bull, Richard J
- Chang, Christine
- Crackett, Peter H
- Deshmukh, Gauri
- Dyke, Hazel J
- Fong, Rina
- Ghilardi, Nico
- Gibbons, Paul
- Hewitt, Peter R
- Johnson, Adam
- Johnson, Tony
- Kenny, Jane R
- Kohli, Pawan Bir
- Kulagowski, Janusz J
- Liimatta, Marya
- Lupardus, Patrick J
- Maxey, Robert J
- Mendonca, Rohan
- Narukulla, Raman
- Pulk, Rebecca
- Ubhayakar, Savita
- van Abbema, Anne
- Ward, Stuart I
- Waszkowycz, Bohdan
- Zak, Mark
Producer: 20140424
In:
Bioorganic & medicinal chemistry letters vol. 23
Availability: No items available.
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8.
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Discovery of a class of highly potent Janus Kinase 1/2 (JAK1/2) inhibitors demonstrating effective cell-based blockade of IL-13 signaling. [electronic resource] by
- Zak, Mark
- Hanan, Emily J
- Lupardus, Patrick
- Brown, David G
- Robinson, Colin
- Siu, Michael
- Lyssikatos, Joseph P
- Romero, F Anthony
- Zhao, Guiling
- Kellar, Terry
- Mendonca, Rohan
- Ray, Nicholas C
- Goodacre, Simon C
- Crackett, Peter H
- McLean, Neville
- Hurley, Christopher A
- Yuen, Po-Wai
- Cheng, Yun-Xing
- Liu, Xiongcai
- Liimatta, Marya
- Kohli, Pawan Bir
- Nonomiya, Jim
- Salmon, Gary
- Buckley, Gerry
- Lloyd, Julia
- Gibbons, Paul
- Ghilardi, Nico
- Kenny, Jane R
- Johnson, Adam
Producer: 20200921
In:
Bioorganic & medicinal chemistry letters vol. 29
Availability: No items available.
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9.
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Identification of C-2 hydroxyethyl imidazopyrrolopyridines as potent JAK1 inhibitors with favorable physicochemical properties and high selectivity over JAK2. [electronic resource] by
- Zak, Mark
- Hurley, Christopher A
- Ward, Stuart I
- Bergeron, Philippe
- Barrett, Kathy
- Balazs, Mercedesz
- Blair, Wade S
- Bull, Richard
- Chakravarty, Paroma
- Chang, Christine
- Crackett, Peter
- Deshmukh, Gauri
- DeVoss, Jason
- Dragovich, Peter S
- Eigenbrot, Charles
- Ellwood, Charles
- Gaines, Simon
- Ghilardi, Nico
- Gibbons, Paul
- Gradl, Stefan
- Gribling, Peter
- Hamman, Chris
- Harstad, Eric
- Hewitt, Peter
- Johnson, Adam
- Johnson, Tony
- Kenny, Jane R
- Koehler, Michael F T
- Bir Kohli, Pawan
- Labadie, Sharada
- Lee, Wyne P
- Liao, Jiangpeng
- Liimatta, Marya
- Mendonca, Rohan
- Narukulla, Raman
- Pulk, Rebecca
- Reeve, Austin
- Savage, Scott
- Shia, Steven
- Steffek, Micah
- Ubhayakar, Savita
- van Abbema, Anne
- Aliagas, Ignacio
- Avitabile-Woo, Barbara
- Xiao, Yisong
- Yang, Jing
- Kulagowski, Janusz J
Producer: 20130820
In:
Journal of medicinal chemistry vol. 56
Availability: No items available.
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