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2-Aryl benzimidazoles featuring alkyl-linked pendant alcohols and amines as inhibitors of checkpoint kinase Chk2. [electronic resource] by
- Neff, Danielle K
- Lee-Dutra, Alice
- Blevitt, Jonathan M
- Axe, Frank U
- Hack, Michael D
- Buma, Johnathan C
- Rynberg, Raymond
- Brunmark, Anders
- Karlsson, Lars
- Breitenbucher, J Guy
Producer: 20080303
In:
Bioorganic & medicinal chemistry letters vol. 17
Availability: No items available.
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9.
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A novel B-RAF inhibitor blocks interleukin-8 (IL-8) synthesis in human melanoma xenografts, revealing IL-8 as a potential pharmacodynamic biomarker. [electronic resource] by
- Crawford, Shelby
- Belajic, Daniel
- Wei, Jianmei
- Riley, Jason P
- Dunford, Paul J
- Bembenek, Scott
- Fourie, Anne
- Edwards, James P
- Karlsson, Lars
- Brunmark, Anders
- Wolin, Ronald L
- Blevitt, Jonathan M
Producer: 20080619
In:
Molecular cancer therapeutics vol. 7
Availability: No items available.
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10.
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Polypharmacology of Small-Molecule Modulators of the 5-Lipoxygenase Activating Protein (FLAP) Observed via a High-throughput Lipidomics Platform. [electronic resource] by
- Song, Jiao
- Liu, Xuejun
- Zhu, Jian
- Tootoonchi, Mandana
- Keith, John M
- Meduna, Steven P
- Dvorak, Curt A
- Eccles, Wendy
- Krawczuk, Paul J
- Blevitt, Jonathan M
- Wu, Jiejun
- Rao, Navin L
- Lebsack, Alec D
- Milla, Marcos E
Producer: 20161014
In:
Journal of biomolecular screening vol. 21
Availability: No items available.
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11.
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Structural Basis of Small-Molecule Aggregate Induced Inhibition of a Protein-Protein Interaction. [electronic resource] by
- Blevitt, Jonathan M
- Hack, Michael D
- Herman, Krystal L
- Jackson, Paul F
- Krawczuk, Paul J
- Lebsack, Alec D
- Liu, Annie X
- Mirzadegan, Taraneh
- Nelen, Marina I
- Patrick, Aaron N
- Steinbacher, Stefan
- Milla, Marcos E
- Lumb, Kevin J
Producer: 20170620
In:
Journal of medicinal chemistry vol. 60
Availability: No items available.
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12.
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Azabenzthiazole inhibitors of leukotriene A₄ hydrolase. [electronic resource] by
- Tanis, Virginia M
- Bacani, Genesis M
- Blevitt, Jonathan M
- Chrovian, Christa C
- Crawford, Shelby
- De Leon, Aimee
- Fourie, Anne M
- Gomez, Laurent
- Grice, Cheryl A
- Herman, Krystal
- Kearney, Aaron M
- Landry-Bayle, Adrienne M
- Lee-Dutra, Alice
- Nelson, Jay
- Riley, Jason P
- Santillán, Alejandro
- Wiener, John J M
- Xue, Xiaohua
- Young, Arlene L
Producer: 20130520
In:
Bioorganic & medicinal chemistry letters vol. 22
Availability: No items available.
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13.
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Identification of benzofuran central cores for the inhibition of leukotriene A(4) hydrolase. [electronic resource] by
- Eccles, Wendy
- Blevitt, Jonathan M
- Booker, Jamila N
- Chrovian, Christa C
- Crawford, Shelby
- de Leon, Aimee Rose
- Deng, Xiaohu
- Fourie, Anne M
- Grice, Cheryl A
- Herman, Krystal
- Karlsson, Lars
- Kearney, Aaron M
- Lee-Dutra, Alice
- Liang, Jimmy
- Luna, Rosa
- Pippel, Dan
- Rao, Navin
- Riley, Jason P
- Santillán, Alejandro
- Savall, Brad
- Tanis, Virginia M
- Xue, Xiaohua
- Young, Arlene L
Producer: 20130625
In:
Bioorganic & medicinal chemistry letters vol. 23
Availability: No items available.
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