Results
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81.
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Potent and selective bicyclic lactam inhibitors of thrombin: Part 2: P1 modifications. [electronic resource] by
- Plummer, J S
- Berryman, K A
- Cai, C
- Cody, W L
- DiMaio, J
- Doherty, A M
- Edmunds, J J
- He, J X
- Holland, D R
- Levesque, S
- Kent, D R
- Narasimhan, L S
- Rubin, J R
- Rapundalo, S T
- Siddiqui, M A
- Susser, A J
- St-Denis, Y
- Winocour, P D
Producer: 19990121
In:
Bioorganic & medicinal chemistry letters vol. 8
Availability: No items available.
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82.
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Synthesis, structure-activity relationships, and pharmacological profile of 9-amino-4-oxo-1-phenyl-3,4,6,7-tetrahydro[1,4]diazepino[6, 7,1-hi]indoles: discovery of potent, selective phosphodiesterase type 4 inhibitors. [electronic resource] by
- Burnouf, C
- Auclair, E
- Avenel, N
- Bertin, B
- Bigot, C
- Calvet, A
- Chan, K
- Durand, C
- Fasquelle, V
- Féru, F
- Gilbertsen, R
- Jacobelli, H
- Kebsi, A
- Lallier, E
- Maignel, J
- Martin, B
- Milano, S
- Ouagued, M
- Pascal, Y
- Pruniaux, M P
- Puaud, J
- Rocher, M N
- Terrasse, C
- Wrigglesworth, R
- Doherty, A M
Producer: 20010118
In:
Journal of medicinal chemistry vol. 43
Availability: No items available.
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83.
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Structure-activity relationships for a novel series of pyrido[2,3-d]pyrimidine tyrosine kinase inhibitors. [electronic resource] by
- Hamby, J M
- Connolly, C J
- Schroeder, M C
- Winters, R T
- Showalter, H D
- Panek, R L
- Major, T C
- Olsewski, B
- Ryan, M J
- Dahring, T
- Lu, G H
- Keiser, J
- Amar, A
- Shen, C
- Kraker, A J
- Slintak, V
- Nelson, J M
- Fry, D W
- Bradford, L
- Hallak, H
- Doherty, A M
Producer: 19970903
In:
Journal of medicinal chemistry vol. 40
Availability: No items available.
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84.
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Synthesis and tyrosine kinase inhibitory activity of a series of 2-amino-8H-pyrido[2,3-d]pyrimidines: identification of potent, selective platelet-derived growth factor receptor tyrosine kinase inhibitors. [electronic resource] by
- Boschelli, D H
- Wu, Z
- Klutchko, S R
- Showalter, H D
- Hamby, J M
- Lu, G H
- Major, T C
- Dahring, T K
- Batley, B
- Panek, R L
- Keiser, J
- Hartl, B G
- Kraker, A J
- Klohs, W D
- Roberts, B J
- Patmore, S
- Elliott, W L
- Steinkampf, R
- Bradford, L A
- Hallak, H
- Doherty, A M
Producer: 19981123
In:
Journal of medicinal chemistry vol. 41
Availability: No items available.
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85.
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Soluble 2-substituted aminopyrido[2,3-d]pyrimidin-7-yl ureas. Structure-activity relationships against selected tyrosine kinases and exploration of in vitro and in vivo anticancer activity. [electronic resource] by
- Schroeder, M C
- Hamby, J M
- Connolly, C J
- Grohar, P J
- Winters, R T
- Barvian, M R
- Moore, C W
- Boushelle, S L
- Crean, S M
- Kraker, A J
- Driscoll, D L
- Vincent, P W
- Elliott, W L
- Lu, G H
- Batley, B L
- Dahring, T K
- Major, T C
- Panek, R L
- Doherty, A M
- Showalter, H D
Producer: 20010628
In:
Journal of medicinal chemistry vol. 44
Availability: No items available.
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86.
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2-Substituted aminopyrido[2,3-d]pyrimidin-7(8H)-ones. structure-activity relationships against selected tyrosine kinases and in vitro and in vivo anticancer activity. [electronic resource] by
- Klutchko, S R
- Hamby, J M
- Boschelli, D H
- Wu, Z
- Kraker, A J
- Amar, A M
- Hartl, B G
- Shen, C
- Klohs, W D
- Steinkampf, R W
- Driscoll, D L
- Nelson, J M
- Elliott, W L
- Roberts, B J
- Stoner, C L
- Vincent, P W
- Dykes, D J
- Panek, R L
- Lu, G H
- Major, T C
- Dahring, T K
- Hallak, H
- Bradford, L A
- Showalter, H D
- Doherty, A M
Producer: 19980909
In:
Journal of medicinal chemistry vol. 41
Availability: No items available.
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