Results
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4861.
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A strong glutathione S-transferase inhibitor overcomes the P-glycoprotein-mediated resistance in tumor cells. 6-(7-Nitro-2,1,3-benzoxadiazol-4-ylthio)hexanol (NBDHEX) triggers a caspase-dependent apoptosis in MDR1-expressing leukemia cells. [electronic resource] by
- Turella, Paola
- Filomeni, Giuseppe
- Dupuis, Maria Luisa
- Ciriolo, Maria Rosa
- Molinari, Agnese
- De Maria, Francesca
- Tombesi, Marina
- Cianfriglia, Maurizio
- Federici, Giorgio
- Ricci, Giorgio
- Caccuri, Anna Maria
Producer: 20060925
In:
The Journal of biological chemistry vol. 281
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4862.
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Discovery of 14-3-3 protein-protein interaction inhibitors that sensitize multidrug-resistant cancer cells to doxorubicin and the Akt inhibitor GSK690693. [electronic resource] by
- Mori, Mattia
- Vignaroli, Giulia
- Cau, Ylenia
- Dinić, Jelena
- Hill, Richard
- Rossi, Matteo
- Colecchia, David
- Pešić, Milica
- Link, Wolfgang
- Chiariello, Mario
- Ottmann, Christian
- Botta, Maurizio
Producer: 20150221
In:
ChemMedChem vol. 9
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4863.
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The development and maintenance of paclitaxel-induced neuropathic pain require activation of the sphingosine 1-phosphate receptor subtype 1. [electronic resource] by
- Janes, Kali
- Little, Joshua W
- Li, Chao
- Bryant, Leesa
- Chen, Collin
- Chen, Zhoumou
- Kamocki, Krzysztof
- Doyle, Timothy
- Snider, Ashley
- Esposito, Emanuela
- Cuzzocrea, Salvatore
- Bieberich, Erhard
- Obeid, Lina
- Petrache, Irina
- Nicol, Grant
- Neumann, William L
- Salvemini, Daniela
Producer: 20150211
In:
The Journal of biological chemistry vol. 289
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4864.
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Ataluren for the treatment of nonsense-mutation cystic fibrosis: a randomised, double-blind, placebo-controlled phase 3 trial. [electronic resource] by
- Kerem, Eitan
- Konstan, Michael W
- De Boeck, Kris
- Accurso, Frank J
- Sermet-Gaudelus, Isabelle
- Wilschanski, Michael
- Elborn, J Stuart
- Melotti, Paola
- Bronsveld, Inez
- Fajac, Isabelle
- Malfroot, Anne
- Rosenbluth, Daniel B
- Walker, Patricia A
- McColley, Susanna A
- Knoop, Christiane
- Quattrucci, Serena
- Rietschel, Ernst
- Zeitlin, Pamela L
- Barth, Jay
- Elfring, Gary L
- Welch, Ellen M
- Branstrom, Arthur
- Spiegel, Robert J
- Peltz, Stuart W
- Ajayi, Temitayo
- Rowe, Steven M
Producer: 20150330
In:
The Lancet. Respiratory medicine vol. 2
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4865.
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4866.
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Discovery and preliminary evaluation of 2-aminobenzamide and hydroxamate derivatives containing 1,2,4-oxadiazole moiety as potent histone deacetylase inhibitors. [electronic resource] by
- Cai, Jin
- Wei, Hongtao
- Hong, Kwon Ho
- Wu, Xiaoqing
- Cao, Meng
- Zong, Xi
- Li, Lushen
- Sun, Chunlong
- Chen, Junqing
- Ji, Min
Producer: 20160216
In:
European journal of medicinal chemistry vol. 96
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4867.
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New potent antibacterials against Gram-positive multiresistant pathogens: effects of side chain modification and chirality in linezolid-like 1,2,4-oxadiazoles. [electronic resource] by
- Fortuna, Cosimo G
- Berardozzi, Roberto
- Bonaccorso, Carmela
- Caltabiano, Gianluigi
- Di Bari, Lorenzo
- Goracci, Laura
- Guarcello, Annalisa
- Pace, Andrea
- Palumbo Piccionello, Antonio
- Pescitelli, Gennaro
- Pierro, Paola
- Lonati, Elena
- Bulbarelli, Alessandra
- Cocuzza, Clementina E A
- Musumarra, Giuseppe
- Musumeci, Rosario
Producer: 20150803
In:
Bioorganic & medicinal chemistry vol. 22
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4868.
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Attenuated methamphetamine-induced locomotor sensitization in serotonin transporter knockout mice is restored by serotonin 1B receptor antagonist treatment. [electronic resource] by
- Igari, Moe
- Shen, Hao-Wei
- Hagino, Yoko
- Fukushima, Setsu
- Kasahara, Yoshiyuki
- Lesch, Klaus-Peter
- Murphy, Dennis L
- Hall, Frank Scott
- Uhl, George R
- Ikeda, Kazutaka
- Yaegashi, Nobuo
- Sora, Ichiro
Producer: 20150903
In:
Behavioural pharmacology vol. 26
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4869.
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Direct angiotensin II type 2 receptor stimulation by compound 21 prevents vascular dementia. [electronic resource] by
- Iwanami, Jun
- Mogi, Masaki
- Tsukuda, Kana
- Wang, Xiao-Li
- Nakaoka, Hirotomo
- Kan-no, Harumi
- Chisaka, Toshiyuki
- Bai, Hui-Yu
- Shan, Bao-Shuai
- Kukida, Masayoshi
- Horiuchi, Masatsugu
Producer: 20160115
In:
Journal of the American Society of Hypertension : JASH vol. 9
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4870.
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4871.
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4872.
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The S1P1 receptor-selective agonist CYM-5442 protects retinal ganglion cells in endothelin-1 induced retinal ganglion cell loss. [electronic resource] by
- Blanco, Román
- Martínez-Navarrete, Gema
- Valiente-Soriano, Francisco J
- Avilés-Trigueros, Marcelino
- Pérez-Rico, Consuelo
- Serrano-Puebla, Ana
- Boya, Patricia
- Fernández, Eduardo
- Vidal-Sanz, Manuel
- de la Villa, Pedro
Producer: 20171012
In:
Experimental eye research vol. 164
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4873.
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4874.
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4875.
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5-Aryl-1,3,4-oxadiazol-2-ylthioalkanoic Acids: A Highly Potent New Class of Inhibitors of Rho/Myocardin-Related Transcription Factor (MRTF)/Serum Response Factor (SRF)-Mediated Gene Transcription as Potential Antifibrotic Agents for Scleroderma. [electronic resource] by
- Kahl, Dylan J
- Hutchings, Kim M
- Lisabeth, Erika Mathes
- Haak, Andrew J
- Leipprandt, Jeffrey R
- Dexheimer, Thomas
- Khanna, Dinesh
- Tsou, Pei-Suen
- Campbell, Phillip L
- Fox, David A
- Wen, Bo
- Sun, Duxin
- Bailie, Marc
- Neubig, Richard R
- Larsen, Scott D
Producer: 20200622
In:
Journal of medicinal chemistry vol. 62
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4876.
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