Results
|
161.
|
Novel fused oxazepino-indoles (FOIs) attenuate liver carcinogenesis via IL-6/JAK2/STAT3 signaling blockade as evidenced through data-based mathematical modeling. [electronic resource] by
- Singh, Ashok K
- Bhadauria, Archana Singh
- Kumar, Umesh
- Raj, Vinit
- Maurya, Vimal
- Kumar, Dinesh
- Maity, Biswanath
- Prakash, Anand
- De, Arnab
- Samanta, Amalesh
- Saha, Sudipta
Producer: 20180523
In:
Life sciences vol. 201
Availability: No items available.
|
|
162.
|
|
|
163.
|
|
|
164.
|
|
|
165.
|
Discovery of Second Generation Reversible Covalent DPP1 Inhibitors Leading to an Oxazepane Amidoacetonitrile Based Clinical Candidate (AZD7986). [electronic resource] by
- Doyle, Kevin
- Lönn, Hans
- Käck, Helena
- Van de Poël, Amanda
- Swallow, Steve
- Gardiner, Philip
- Connolly, Stephen
- Root, James
- Wikell, Cecilia
- Dahl, Göran
- Stenvall, Kristina
- Johannesson, Petra
Producer: 20170606
In:
Journal of medicinal chemistry vol. 59
Availability: No items available.
|
|
166.
|
Discovery and development of benzo-[1,2,4]-triazolo-[1,4]-oxazepine GPR142 agonists for the treatment of diabetes. [electronic resource] by
- Wilson, Jonathan E
- Kurukulasuriya, Ravi
- Sinz, Christopher
- Lombardo, Matthew
- Bender, Kate
- Parker, Dann
- Sherer, Edward C
- Costa, Melissa
- Dingley, Karen
- Li, Xiaofang
- Mitelman, Stanley
- Tong, Sharon
- Bugianesi, Randal
- Ehrhardt, Anka
- Priest, Birgit
- Ratliff, Kevin
- Ujjainwalla, Feroze
- Nargund, Ravi
- Hagmann, William K
- Edmondson, Scott
Producer: 20170720
In:
Bioorganic & medicinal chemistry letters vol. 26
Availability: No items available.
|
|
167.
|
The pyrrolo-1,5-benzoxazepine, PBOX-6, inhibits the growth of breast cancer cells in vitro independent of estrogen receptor status and inhibits breast tumour growth in vivo. [electronic resource] by
- Greene, Lisa M
- Fleeton, Marina
- Mulligan, Jude
- Gowda, Chikkanna
- Sheahan, Brian J
- Atkins, Gregory J
- Campiani, Giuseppe
- Nacci, Vito
- Lawler, Mark
- Williams, D Clive
- Zisterer, Daniela M
Producer: 20051114
In:
Oncology reports vol. 14
Availability: No items available.
|
|
168.
|
Enantioselective binding of second generation pyrrolobenzoxazepinones to the catalytic ternary complex of HIV-1 RT wild-type and L100I and K103N drug resistant mutants. [electronic resource] by
- Butini, Stefania
- Gemma, Sandra
- Brindisi, Margherita
- Borrelli, Giuseppe
- Fiorini, Isabella
- Samuele, Alberta
- Karytinos, Aristotele
- Facchini, Marcella
- Lossani, Andrea
- Zanoli, Samantha
- Campiani, Giuseppe
- Novellino, Ettore
- Focher, Federico
- Maga, Giovanni
Producer: 20111122
In:
Bioorganic & medicinal chemistry letters vol. 21
Availability: No items available.
|
|
169.
|
|
|
170.
|
|
|
171.
|
|
|
172.
|
|
|
173.
|
Benzoxazepines Achieve Potent Suppression of IL-17 Release in Human T-Helper 17 (TH 17) Cells through an Induced-Fit Binding Mode to the Nuclear Receptor RORγ. [electronic resource] by
- Olsson, Roine I
- Xue, Yafeng
- von Berg, Stefan
- Aagaard, Anna
- McPheat, Jane
- Hansson, Eva L
- Bernström, Jenny
- Hansson, Pia
- Jirholt, Johan
- Grindebacke, Hanna
- Leffler, Agnes
- Chen, Rongfeng
- Xiong, Yao
- Ge, Hongbin
- Hansson, Thomas G
- Narjes, Frank
Producer: 20160919
In:
ChemMedChem vol. 11
Availability: No items available.
|
|
174.
|
|
|
175.
|
Dibenzo[b,f][1,4]oxazepines and dibenzo[b,e]oxepines: Influence of the chlorine substitution pattern on the pharmacology at the H [electronic resource] by
- Naporra, Franziska
- Gobleder, Susanne
- Wittmann, Hans-Joachim
- Spindler, Julia
- Bodensteiner, Michael
- Bernhardt, Günther
- Hübner, Harald
- Gmeiner, Peter
- Elz, Sigurd
- Strasser, Andrea
Producer: 20171218
In:
Pharmacological research vol. 113
Availability: No items available.
|
|
176.
|
|
|
177.
|
Defining the key pharmacophore elements of PF-04620110: discovery of a potent, orally-active, neutral DGAT-1 inhibitor. [electronic resource] by
- Dow, Robert L
- Andrews, Melissa P
- Li, Jian-Cheng
- Michael Gibbs, E
- Guzman-Perez, Angel
- Laperle, Jennifer L
- Li, Qifang
- Mather, Dawn
- Munchhof, Michael J
- Niosi, Mark
- Patel, Leena
- Perreault, Christian
- Tapley, Susan
- Zavadoski, William J
Producer: 20140318
In:
Bioorganic & medicinal chemistry vol. 21
Availability: No items available.
|
|
178.
|
Microtubule-targeting-compound PBOX-15 radiosensitizes cancer cells in vitro. [electronic resource] by
- Forde, James C
- Maginn, Elaina N
- McNamara, Gillian
- Martin, Lynn M
- Campiani, Guiseppe
- Williams, D Clive
- Zisterer, Daniela
- McElligott, Anthony M
- Lawler, Mark
- Lynch, Thomas H
- Hollywood, Donal
- Marignol, Laure
Producer: 20110614
In:
Cancer biology & therapy vol. 11
Availability: No items available.
|
|
179.
|
|
|
180.
|
|