Inhibition of cruzipain visualized in a fluorescence quenched solid-phase inhibitor library assay. D-amino acid inhibitors for cruzipain, cathepsin B and cathepsin L. [electronic resource]
Producer: 19980806Description: 83-91 p. digitalISSN:- 1075-2617
- Amino Acids -- pharmacology
- Animals
- Binding Sites -- physiology
- Binding, Competitive
- Cathepsin B -- metabolism
- Cathepsin L
- Cathepsins -- metabolism
- Cysteine Endopeptidases -- metabolism
- Endopeptidases
- Enzyme Inhibitors -- pharmacology
- Fluorescent Dyes -- metabolism
- Humans
- Kallikreins -- metabolism
- Kinetics
- Mammals
- Models, Molecular
- Peptide Library
- Peptides -- chemical synthesis
- Protein Conformation
- Protozoan Proteins -- metabolism
- Substrate Specificity
- Trypanosoma cruzi -- enzymology
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Publication Type: Journal Article; Research Support, Non-U.S. Gov't
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