Synthesis and opioid antagonist potencies of naltrexamine bivalent ligands with conformationally restricted spacers. [electronic resource]
Producer: 19861022Description: 1650-3 p. digitalISSN:- 0022-2623
- Animals
- Biological Assay
- Chemical Phenomena
- Chemistry
- Cyclazocine -- analogs & derivatives
- Endorphins -- antagonists & inhibitors
- Ethylketocyclazocine
- Guinea Pigs
- Ileum -- physiology
- Molecular Conformation
- Morphine -- pharmacology
- Muscle Contraction -- drug effects
- Naltrexone -- analogs & derivatives
- Receptors, Opioid -- drug effects
- Receptors, Opioid, kappa
- Receptors, Opioid, mu
- Structure-Activity Relationship
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Publication Type: Journal Article; Research Support, U.S. Gov't, P.H.S.
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