Inactivation of PP2A by a recurrent mutation drives resistance to MEK inhibitors. [electronic resource]
Producer: 20200619Description: 703-717 p. digitalISSN:- 1476-5594
- Amino Acid Substitution
- Arginine -- genetics
- Calmodulin-Binding Proteins -- metabolism
- Carcinogenesis -- drug effects
- Cell Line, Tumor
- Drug Resistance, Neoplasm -- genetics
- Humans
- MAP Kinase Signaling System -- drug effects
- Membrane Proteins -- metabolism
- Mitogen-Activated Protein Kinase Kinases -- antagonists & inhibitors
- Molecular Dynamics Simulation
- Mutagenesis, Site-Directed
- Mutation
- Neoplasms -- drug therapy
- Nerve Tissue Proteins -- metabolism
- Protein Kinase Inhibitors -- pharmacology
- Protein Phosphatase 2 -- genetics
- Recombinant Proteins -- genetics
- Transfection
- Tyrosine -- genetics
- Xenograft Model Antitumor Assays
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Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't
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