Cyclization-blocked proguanil as a strategy to improve the antimalarial activity of atovaquone. [electronic resource]
Producer: 20200420Description: 166 p. digitalISSN:- 2399-3642
- Animals
- Anopheles
- Antimalarials -- chemistry
- Atovaquone -- chemistry
- Cyclization -- drug effects
- Dihydroorotate Dehydrogenase
- Dose-Response Relationship, Drug
- Drug Combinations
- Electron Transport Complex III -- antagonists & inhibitors
- Enzyme Inhibitors -- chemistry
- Erythrocytes -- drug effects
- Folic Acid -- metabolism
- Hep G2 Cells
- Humans
- Inhibitory Concentration 50
- Liver -- drug effects
- Oxidoreductases Acting on CH-CH Group Donors -- metabolism
- Plasmodium berghei -- drug effects
- Plasmodium falciparum -- drug effects
- Proguanil -- analogs & derivatives
- Sporozoites -- drug effects
- Terpenes -- metabolism
- Triazines -- chemistry
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Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't
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