Discovery and Characterization of the Potent and Highly Selective (Piperidin-4-yl)pyrido[3,2- d]pyrimidine Based in Vitro Probe BAY-885 for the Kinase ERK5. [electronic resource]
Producer: 20191017Description: 928-940 p. digitalISSN:- 1520-4804
- Apoptosis -- drug effects
- Binding Sites
- Cell Differentiation -- drug effects
- Cell Line
- Cell Proliferation -- drug effects
- Crystallography, X-Ray
- Drug Evaluation, Preclinical
- Half-Life
- Humans
- Mitogen-Activated Protein Kinase 7 -- antagonists & inhibitors
- Molecular Docking Simulation
- Protein Kinase Inhibitors -- chemistry
- Protein Structure, Tertiary
- Pyridines -- chemistry
- Pyrimidines -- chemistry
- Signal Transduction -- drug effects
- Structure-Activity Relationship
- Transcription, Genetic -- drug effects
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Publication Type: Journal Article
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