Discovery of GDC-0853: A Potent, Selective, and Noncovalent Bruton's Tyrosine Kinase Inhibitor in Early Clinical Development. [electronic resource]
Producer: 20190417Description: 2227-2245 p. digitalISSN:- 1520-4804
- Agammaglobulinaemia Tyrosine Kinase -- antagonists & inhibitors
- Animals
- Anti-Inflammatory Agents -- pharmacokinetics
- Arthritis, Experimental -- drug therapy
- Arthritis, Rheumatoid -- drug therapy
- Dogs
- Drug Discovery
- Humans
- Lupus Erythematosus, Systemic -- drug therapy
- Madin Darby Canine Kidney Cells
- Models, Molecular
- Molecular Structure
- Piperazines -- pharmacokinetics
- Protein Kinase Inhibitors -- pharmacokinetics
- Pyridones -- pharmacokinetics
- Rats
- Rats, Inbred Lew
- Rats, Sprague-Dawley
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Publication Type: Journal Article
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