Discovery of GDC-0853: A Potent, Selective, and Noncovalent Bruton's Tyrosine Kinase Inhibitor in Early Clinical Development. (Record no. 28100127)
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| 000 -LEADER | |
|---|---|
| fixed length control field | 02299 a2200697 4500 |
| 005 - DATE AND TIME OF LATEST TRANSACTION | |
| control field | 20250517202219.0 |
| 008 - FIXED-LENGTH DATA ELEMENTS--GENERAL INFORMATION | |
| fixed length control field | 201904s 0 0 eng d |
| 022 ## - INTERNATIONAL STANDARD SERIAL NUMBER | |
| International Standard Serial Number | 1520-4804 |
| 024 7# - OTHER STANDARD IDENTIFIER | |
| Standard number or code | 10.1021/acs.jmedchem.7b01712 |
| Source of number or code | doi |
| 040 ## - CATALOGING SOURCE | |
| Original cataloging agency | NLM |
| Language of cataloging | eng |
| Transcribing agency | NLM |
| 100 1# - MAIN ENTRY--PERSONAL NAME | |
| Personal name | Crawford, James J |
| 264 #0 - PRODUCTION, PUBLICATION, DISTRIBUTION, MANUFACTURE, AND COPYRIGHT NOTICE | |
| Date of production, publication, distribution, manufacture, or copyright notice | 20190417 |
| 245 00 - TITLE STATEMENT | |
| Title | Discovery of GDC-0853: A Potent, Selective, and Noncovalent Bruton's Tyrosine Kinase Inhibitor in Early Clinical Development. |
| Medium | [electronic resource] |
| 260 ## - PUBLICATION, DISTRIBUTION, ETC. | |
| Name of publisher, distributor, etc. | Journal of medicinal chemistry |
| Date of publication, distribution, etc. | 03 2018 |
| 300 ## - PHYSICAL DESCRIPTION | |
| Extent | 2227-2245 p. |
| Other physical details | digital |
| 500 ## - GENERAL NOTE | |
| General note | Publication Type: Journal Article |
| 650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
| Topical term or geographic name entry element | Agammaglobulinaemia Tyrosine Kinase |
| General subdivision | antagonists & inhibitors |
| 650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
| Topical term or geographic name entry element | Animals |
| 650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
| Topical term or geographic name entry element | Anti-Inflammatory Agents |
| General subdivision | pharmacokinetics |
| 650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
| Topical term or geographic name entry element | Arthritis, Experimental |
| General subdivision | drug therapy |
| 650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
| Topical term or geographic name entry element | Arthritis, Rheumatoid |
| General subdivision | drug therapy |
| 650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
| Topical term or geographic name entry element | Dogs |
| 650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
| Topical term or geographic name entry element | Drug Discovery |
| 650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
| Topical term or geographic name entry element | Humans |
| 650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
| Topical term or geographic name entry element | Lupus Erythematosus, Systemic |
| General subdivision | drug therapy |
| 650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
| Topical term or geographic name entry element | Madin Darby Canine Kidney Cells |
| 650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
| Topical term or geographic name entry element | Models, Molecular |
| 650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
| Topical term or geographic name entry element | Molecular Structure |
| 650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
| Topical term or geographic name entry element | Piperazines |
| General subdivision | pharmacokinetics |
| 650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
| Topical term or geographic name entry element | Protein Kinase Inhibitors |
| General subdivision | pharmacokinetics |
| 650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
| Topical term or geographic name entry element | Pyridones |
| General subdivision | pharmacokinetics |
| 650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
| Topical term or geographic name entry element | Rats |
| 650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
| Topical term or geographic name entry element | Rats, Inbred Lew |
| 650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
| Topical term or geographic name entry element | Rats, Sprague-Dawley |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Johnson, Adam R |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Misner, Dinah L |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Belmont, Lisa D |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Castanedo, Georgette |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Choy, Regina |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Coraggio, Melis |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Dong, Liming |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Eigenbrot, Charles |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Erickson, Rebecca |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Ghilardi, Nico |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Hau, Jonathan |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Katewa, Arna |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Kohli, Pawan Bir |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Lee, Wendy |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Lubach, Joseph W |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | McKenzie, Brent S |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Ortwine, Daniel F |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Schutt, Leah |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Tay, Suzanne |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Wei, BinQing |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Reif, Karin |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Liu, Lichuan |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Wong, Harvey |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Young, Wendy B |
| 773 0# - HOST ITEM ENTRY | |
| Title | Journal of medicinal chemistry |
| Related parts | vol. 61 |
| -- | no. 6 |
| -- | p. 2227-2245 |
| 856 40 - ELECTRONIC LOCATION AND ACCESS | |
| Uniform Resource Identifier | <a href="https://doi.org/10.1021/acs.jmedchem.7b01712">https://doi.org/10.1021/acs.jmedchem.7b01712</a> |
| Public note | Available from publisher's website |
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