Structure-based development of novel triazoles and related thiazolotriazoles as anticancer agents and Cdc25A/B phosphatase inhibitors. Synthesis, in vitro biological evaluation, molecular docking and in silico ADME-T studies. [electronic resource]
Producer: 20171018Description: 263-279 p. digitalISSN:- 1768-3254
- Antineoplastic Agents -- chemical synthesis
- Cell Line, Tumor
- Cell Proliferation -- drug effects
- Dose-Response Relationship, Drug
- Drug Screening Assays, Antitumor
- Enzyme Inhibitors -- chemical synthesis
- Humans
- Molecular Docking Simulation
- Molecular Structure
- Structure-Activity Relationship
- Triazoles -- chemical synthesis
- cdc25 Phosphatases -- antagonists & inhibitors
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Publication Type: Journal Article
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