Structure-based development of novel triazoles and related thiazolotriazoles as anticancer agents and Cdc25A/B phosphatase inhibitors. Synthesis, in vitro biological evaluation, molecular docking and in silico ADME-T studies.
Rostom, Sherif A F
Structure-based development of novel triazoles and related thiazolotriazoles as anticancer agents and Cdc25A/B phosphatase inhibitors. Synthesis, in vitro biological evaluation, molecular docking and in silico ADME-T studies. [electronic resource] - European journal of medicinal chemistry Oct 2017 - 263-279 p. digital
Publication Type: Journal Article
1768-3254
10.1016/j.ejmech.2017.07.053 doi
Antineoplastic Agents--chemical synthesis
Cell Line, Tumor
Cell Proliferation--drug effects
Dose-Response Relationship, Drug
Drug Screening Assays, Antitumor
Enzyme Inhibitors--chemical synthesis
Humans
Molecular Docking Simulation
Molecular Structure
Structure-Activity Relationship
Triazoles--chemical synthesis
cdc25 Phosphatases--antagonists & inhibitors
Structure-based development of novel triazoles and related thiazolotriazoles as anticancer agents and Cdc25A/B phosphatase inhibitors. Synthesis, in vitro biological evaluation, molecular docking and in silico ADME-T studies. [electronic resource] - European journal of medicinal chemistry Oct 2017 - 263-279 p. digital
Publication Type: Journal Article
1768-3254
10.1016/j.ejmech.2017.07.053 doi
Antineoplastic Agents--chemical synthesis
Cell Line, Tumor
Cell Proliferation--drug effects
Dose-Response Relationship, Drug
Drug Screening Assays, Antitumor
Enzyme Inhibitors--chemical synthesis
Humans
Molecular Docking Simulation
Molecular Structure
Structure-Activity Relationship
Triazoles--chemical synthesis
cdc25 Phosphatases--antagonists & inhibitors