Inhibiting fungal multidrug resistance by disrupting an activator-Mediator interaction. [electronic resource]
Producer: 20160315Description: 485-9 p. digitalISSN:- 1476-4687
- Animals
- Antifungal Agents -- pharmacology
- Binding Sites -- drug effects
- Candida glabrata -- drug effects
- Candidiasis -- drug therapy
- DNA-Binding Proteins -- genetics
- Drug Resistance, Fungal -- drug effects
- Drug Resistance, Multiple, Fungal -- drug effects
- Fluconazole -- pharmacology
- Fungal Proteins -- metabolism
- Gene Expression Regulation, Fungal -- drug effects
- Hydrazines -- pharmacokinetics
- Ketoconazole -- pharmacology
- Mediator Complex -- chemistry
- Mice
- Models, Molecular
- Nuclear Magnetic Resonance, Biomolecular
- Protein Binding -- drug effects
- Protein Structure, Tertiary
- Saccharomyces cerevisiae Proteins -- chemistry
- Thiourea -- analogs & derivatives
- Trans-Activators -- chemistry
- Transcription Factors -- genetics
- Transcriptional Activation -- drug effects
- Up-Regulation -- drug effects
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Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't
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