Structure- and function-based design of Plasmodium-selective proteasome inhibitors. [electronic resource]
Producer: 20160224Description: 233-6 p. digitalISSN:- 1476-4687
- Animals
- Antimalarials -- adverse effects
- Artemisinins -- pharmacology
- Catalytic Domain
- Cryoelectron Microscopy
- Dose-Response Relationship, Drug
- Drug Design
- Drug Resistance
- Drug Synergism
- Enzyme Activation
- Female
- Humans
- Mice
- Mice, Inbred BALB C
- Models, Molecular
- Plasmodium -- drug effects
- Plasmodium chabaudi -- drug effects
- Plasmodium falciparum -- drug effects
- Proteasome Endopeptidase Complex -- chemistry
- Proteasome Inhibitors -- adverse effects
- Protein Subunits -- antagonists & inhibitors
- Species Specificity
- Substrate Specificity -- drug effects
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Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't
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