The plasticizer BBP selectively inhibits epigenetic regulator sirtuins. [electronic resource]
Producer: 20160307Description: 130-41 p. digitalISSN:- 1879-3185
- Binding Sites
- Crystallography
- Dose-Response Relationship, Drug
- Endocrine Disruptors -- metabolism
- Epigenesis, Genetic -- drug effects
- Gene Expression Regulation
- Hep G2 Cells
- Hepatocytes -- drug effects
- Histone Deacetylase Inhibitors -- metabolism
- Humans
- Hydrogen Bonding
- Ligands
- Mitochondria, Liver -- drug effects
- Molecular Docking Simulation
- NF-E2-Related Factor 2 -- genetics
- Nuclear Respiratory Factor 1 -- genetics
- Organelle Biogenesis
- Peroxisome Proliferator-Activated Receptor Gamma Coactivator 1-alpha
- Phthalic Acids -- metabolism
- Plasticizers -- metabolism
- Protein Binding
- Protein Conformation
- RNA Interference
- Reactive Oxygen Species -- metabolism
- Sirtuin 1 -- antagonists & inhibitors
- Sirtuin 3 -- antagonists & inhibitors
- Transcription Factors -- genetics
- Transfection
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Publication Type: Journal Article; Research Support, Non-U.S. Gov't
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