Structure-Based Design and Optimization of Multitarget-Directed 2H-Chromen-2-one Derivatives as Potent Inhibitors of Monoamine Oxidase B and Cholinesterases. [electronic resource]
Producer: 20151012Description: 5561-78 p. digitalISSN:- 1520-4804
- Animals
- Blood-Brain Barrier -- metabolism
- Cholinesterase Inhibitors -- chemistry
- Cholinesterases -- chemistry
- Coumarins -- chemistry
- Dogs
- Drug Design
- Humans
- Inhibitory Concentration 50
- Madin Darby Canine Kidney Cells
- Molecular Docking Simulation
- Monoamine Oxidase -- chemistry
- Monoamine Oxidase Inhibitors -- chemistry
- Permeability
- Protein Conformation
- Rats
- Structure-Activity Relationship
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Publication Type: Journal Article; Research Support, Non-U.S. Gov't
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