Azole antifungal inhibition of buprenorphine, methadone and oxycodone in vitro metabolism. [electronic resource]
Producer: 20160212Description: 374-86 p. digitalISSN:- 1945-2403
- Administration, Oral
- Analgesics, Opioid -- metabolism
- Antifungal Agents -- administration & dosage
- Azoles -- administration & dosage
- Biotransformation
- Buprenorphine -- metabolism
- Chromatography, Liquid
- Cytochrome P-450 Enzyme Inhibitors -- administration & dosage
- Cytochrome P-450 Enzyme System -- metabolism
- Dose-Response Relationship, Drug
- Drug Interactions
- Humans
- Isoenzymes
- Kinetics
- Liver -- drug effects
- Methadone -- metabolism
- Microsomes, Liver -- drug effects
- Models, Biological
- Molecular Structure
- Oxycodone -- metabolism
- Recombinant Proteins -- metabolism
- Risk Assessment
- Spectrometry, Mass, Electrospray Ionization
- Structure-Activity Relationship
- Substrate Specificity
- Tandem Mass Spectrometry
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Publication Type: Comparative Study; Journal Article; Research Support, U.S. Gov't, Non-P.H.S.
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