Afatinib circumvents multidrug resistance via dually inhibiting ATP binding cassette subfamily G member 2 in vitro and in vivo. [electronic resource]
Producer: 20151020Description: 11971-85 p. digitalISSN:- 1949-2553
- ATP Binding Cassette Transporter, Subfamily G, Member 2
- ATP-Binding Cassette Transporters -- antagonists & inhibitors
- Afatinib
- Animals
- Antineoplastic Agents -- pharmacology
- Blotting, Western
- Cell Line, Tumor
- Drug Resistance, Multiple -- drug effects
- Drug Resistance, Neoplasm -- drug effects
- Female
- Flow Cytometry
- Humans
- Immunohistochemistry
- In Vitro Techniques
- Male
- Mice
- Mice, Inbred BALB C
- Neoplasm Proteins -- antagonists & inhibitors
- Neoplasms, Experimental -- drug therapy
- Quinazolines -- pharmacology
- Real-Time Polymerase Chain Reaction
- Topotecan -- pharmacology
- Xenograft Model Antitumor Assays
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Publication Type: Journal Article; Research Support, Non-U.S. Gov't
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