Afatinib circumvents multidrug resistance via dually inhibiting ATP binding cassette subfamily G member 2 in vitro and in vivo.
Wang, Xiao-Kun
Afatinib circumvents multidrug resistance via dually inhibiting ATP binding cassette subfamily G member 2 in vitro and in vivo. [electronic resource] - Oncotarget Dec 2014 - 11971-85 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1949-2553
10.18632/oncotarget.2647 doi
ATP Binding Cassette Transporter, Subfamily G, Member 2
ATP-Binding Cassette Transporters--antagonists & inhibitors
Afatinib
Animals
Antineoplastic Agents--pharmacology
Blotting, Western
Cell Line, Tumor
Drug Resistance, Multiple--drug effects
Drug Resistance, Neoplasm--drug effects
Female
Flow Cytometry
Humans
Immunohistochemistry
In Vitro Techniques
Male
Mice
Mice, Inbred BALB C
Neoplasm Proteins--antagonists & inhibitors
Neoplasms, Experimental--drug therapy
Quinazolines--pharmacology
Real-Time Polymerase Chain Reaction
Topotecan--pharmacology
Xenograft Model Antitumor Assays
Afatinib circumvents multidrug resistance via dually inhibiting ATP binding cassette subfamily G member 2 in vitro and in vivo. [electronic resource] - Oncotarget Dec 2014 - 11971-85 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1949-2553
10.18632/oncotarget.2647 doi
ATP Binding Cassette Transporter, Subfamily G, Member 2
ATP-Binding Cassette Transporters--antagonists & inhibitors
Afatinib
Animals
Antineoplastic Agents--pharmacology
Blotting, Western
Cell Line, Tumor
Drug Resistance, Multiple--drug effects
Drug Resistance, Neoplasm--drug effects
Female
Flow Cytometry
Humans
Immunohistochemistry
In Vitro Techniques
Male
Mice
Mice, Inbred BALB C
Neoplasm Proteins--antagonists & inhibitors
Neoplasms, Experimental--drug therapy
Quinazolines--pharmacology
Real-Time Polymerase Chain Reaction
Topotecan--pharmacology
Xenograft Model Antitumor Assays