Mapping the binding pocket of a novel, high-affinity, slow dissociating tachykinin NK3 receptor antagonist: biochemical and electrophysiological characterization. [electronic resource]
Producer: 20150714Description: 259-72 p. digitalISSN:- 1873-7064
- Amino Acid Sequence
- Animals
- Antipsychotic Agents -- pharmacology
- Binding Sites
- Carbamates -- pharmacokinetics
- Central Nervous System Agents -- pharmacology
- Dopaminergic Neurons -- drug effects
- Female
- Gerbillinae
- Guinea Pigs
- HEK293 Cells
- Humans
- Locomotion -- drug effects
- Male
- Models, Molecular
- Molecular Sequence Data
- Mutation
- Neurotransmitter Agents -- pharmacokinetics
- Pars Compacta -- drug effects
- Peptide Fragments -- pharmacology
- Piperidines -- pharmacokinetics
- Receptors, Neurokinin-2 -- antagonists & inhibitors
- Receptors, Neurokinin-3 -- agonists
- Substance P -- analogs & derivatives
- Tissue Culture Techniques
No physical items for this record
Publication Type: Journal Article
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