Mapping the binding pocket of a novel, high-affinity, slow dissociating tachykinin NK3 receptor antagonist: biochemical and electrophysiological characterization.
Malherbe, Pari
Mapping the binding pocket of a novel, high-affinity, slow dissociating tachykinin NK3 receptor antagonist: biochemical and electrophysiological characterization. [electronic resource] - Neuropharmacology Nov 2014 - 259-72 p. digital
Publication Type: Journal Article
1873-7064
10.1016/j.neuropharm.2014.07.017 doi
Amino Acid Sequence
Animals
Antipsychotic Agents--pharmacology
Binding Sites
Carbamates--pharmacokinetics
Central Nervous System Agents--pharmacology
Dopaminergic Neurons--drug effects
Female
Gerbillinae
Guinea Pigs
HEK293 Cells
Humans
Locomotion--drug effects
Male
Models, Molecular
Molecular Sequence Data
Mutation
Neurotransmitter Agents--pharmacokinetics
Pars Compacta--drug effects
Peptide Fragments--pharmacology
Piperidines--pharmacokinetics
Receptors, Neurokinin-2--antagonists & inhibitors
Receptors, Neurokinin-3--agonists
Substance P--analogs & derivatives
Tissue Culture Techniques
Mapping the binding pocket of a novel, high-affinity, slow dissociating tachykinin NK3 receptor antagonist: biochemical and electrophysiological characterization. [electronic resource] - Neuropharmacology Nov 2014 - 259-72 p. digital
Publication Type: Journal Article
1873-7064
10.1016/j.neuropharm.2014.07.017 doi
Amino Acid Sequence
Animals
Antipsychotic Agents--pharmacology
Binding Sites
Carbamates--pharmacokinetics
Central Nervous System Agents--pharmacology
Dopaminergic Neurons--drug effects
Female
Gerbillinae
Guinea Pigs
HEK293 Cells
Humans
Locomotion--drug effects
Male
Models, Molecular
Molecular Sequence Data
Mutation
Neurotransmitter Agents--pharmacokinetics
Pars Compacta--drug effects
Peptide Fragments--pharmacology
Piperidines--pharmacokinetics
Receptors, Neurokinin-2--antagonists & inhibitors
Receptors, Neurokinin-3--agonists
Substance P--analogs & derivatives
Tissue Culture Techniques