Ketoconazole inhibits the cellular uptake of anandamide via inhibition of FAAH at pharmacologically relevant concentrations. [electronic resource]
Producer: 20140929Description: e87542 p. digitalISSN:- 1932-6203
- Amidohydrolases -- antagonists & inhibitors
- Analysis of Variance
- Arachidonic Acids -- metabolism
- Caco-2 Cells
- Dose-Response Relationship, Drug
- Endocannabinoids -- metabolism
- Hep G2 Cells
- Humans
- Ketoconazole -- pharmacology
- Polyunsaturated Alkamides -- metabolism
- Receptor, Cannabinoid, CB2 -- metabolism
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Publication Type: Journal Article; Research Support, Non-U.S. Gov't
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